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2-{1-[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]piperidin-2-yl}acetamide
N-phenyl-5-[2-(1H-pyrazol-1-yl)butanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-6-fluoroquinolin-4-ol
5-cyclopropanecarbonyl-1'-[(6-methylpyridin-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(1H-pyrazol-1-yl)acetamide
4-({4-[3-(1,2,3,6-tetrahydropyridine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
2-[methyl(2-phenylethyl)amino]-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
(1S,5R)-3-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(furan-2-yl)-2-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]formamido}propanoic acid
1-(2,3-difluoro-6-methoxybenzoyl)-4-(1-methylpiperidin-4-yl)piperidine
8-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
ethyl 4-[(4-chlorophenyl)methyl]-1-(quinoxaline-6-carbonyl)piperidine-4-carboxylate
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[4-(methoxymethyl)piperidin-1-yl]methyl}piperidin-2-one
ethyl 4-{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
N-{2-[(6-methoxypyrimidin-4-yl)amino]ethyl}-N-methylmethanesulfonamide
N-(cyclopropylmethyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-(2-chloro-4-{[4-(3-hydroxyphenyl)piperidin-1-yl]methyl}phenoxy)acetamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
2-amino-7-[2-(phenylamino)pyrimidine-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(furan-3-ylmethyl)-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
(3S,4R)-4-(2-methylphenyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidine-3-carboxylic acid
[(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl](methyl)(pyridin-4-ylmethyl)amine
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
6-methyl-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
2-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-1,3-thiazole
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2,6-dimethylquinoline-4-carboxamide
(1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)methanol
[(3R,4R)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(4-chlorophenyl)methyl]-N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-methylpropyl)pyrrolidin-3-yl]pyridine-3-carboxamide
1-(2-fluorophenyl)-4-[6-phenyl-2-(pyrrolidin-1-yl)pyridine-3-carbonyl]piperazine
3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)benzene-1-sulfonamide
1-(1-methanesulfonylpyrrolidine-2-carbonyl)-4-(2-phenoxyethyl)piperazine
3-{2-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}-4-(pyridin-3-ylmethyl)piperazin-2-one
3-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
(3S)-1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}piperidine-3-carboxylic acid
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
5-{[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
(5S,9aS,9bS)-5-(5-cyclopentylthiophen-2-yl)-2-(1-methylpiperidin-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3S,4R)-4-(3-methoxyphenyl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
2,3-dimethyl-7-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-(methylsulfanyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[3-(1H-pyrazol-5-yl)phenyl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxamide
2-[(2R)-2-aminopropanoyl]-N-(cyclopropylmethyl)-N-propyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2,6-dimethylquinoline-4-carboxamide
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
(3S)-3-ethyl-4-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]morpholine
1-(4-methoxyphenyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopropane-1-carboxamide