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5-(hydroxymethyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]furan-2-carboxamide
1-[1-(hydroxymethyl)-9-[(4-methyl-1H-imidazol-2-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-(pyridin-3-yl)ethan-1-one
(2S,4S)-4-[(adamantan-2-yl)amino]-N-ethyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
propyl (4aR,7aS)-4-[(2-methoxyphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
5-ethyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-N-[3-(1,3-oxazol-5-yl)phenyl]piperidine-1-carboxamide
(3R,5S)-N3-methyl-N3-[(1-methyl-1H-imidazol-2-yl)methyl]-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
N1-phenyl-N2-[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]ethane-1,2-diamine
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-5-oxopyrrolidine-3-carboxylic acid
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]propanamide
1-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrrolidine-2-carboxamide
3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
2-[4-(2-aminopyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-benzyl-1H-pyrazol-3-yl)acetamide
4-(cyclohex-3-en-1-ylmethyl)-9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl N-[4-(3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamido)phenyl]carbamate
3-methyl-6-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-3-yl)pyridazine
(2S,4R)-1-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-N-cycloheptyl-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1'-(3-fluorobenzoyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
(1-methyl-5-{[3-(2-methylphenyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
1-(2,3-dihydro-1H-inden-2-yl)-4-(2-ethylpyrimidine-5-carbonyl)-1,4-diazepane
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(propan-2-yl)acetamide
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-[(3-methoxyphenyl)amino]butanamide
2-{3-[3-(6-methoxypyrimidin-4-yl)phenyl]-1H-pyrazol-1-yl}-N,N-dimethylacetamide
2-(5-acetylthiophen-3-yl)-1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]ethan-1-one
4-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2-(trifluoromethyl)morpholine
(2-{1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}ethyl)dimethylamine
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]urea
8-methoxy-2-(2-methoxypyridin-3-yl)quinoline
1-[(2,3-difluorophenyl)methyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-(2H-1,3-benzodioxol-5-yl)-1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-amine
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
N-butyl-N-(furan-2-ylmethyl)-2-(phenylamino)pyrimidine-5-carboxamide
N-{1-[1-(3-phenoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-5-propylthiophene-3-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N'-(4-methylphenyl)-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]propanediamide
1-(2-ethoxyethyl)-5-(4-fluoropiperidine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-[4-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenyl]-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
1-(2-cyclohexylethyl)-3-hydroxy-3-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)piperidin-2-one
(1R,9aR)-1-({[(6-chloropyridin-3-yl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
N-{2-[2-(2,1,3-benzothiadiazol-5-yl)-1H-imidazol-1-yl]ethyl}acetamide
(3S,4R)-1-{imidazo[1,2-a]pyridine-2-carbonyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(1H-imidazole-5-carbonyl)piperidine
N-(1,4-dioxan-2-ylmethyl)-N-methyl-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(2-methoxyethyl)methylamine
N4-(4-cyano-2-ethylphenyl)morpholine-2,4-dicarboxamide
(3S)-1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylazepan-3-amine