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5-chloro-2-{2-[2-(2-methyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
1-(4-fluorophenyl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrrolidin-3-amine
3-(pentan-2-yl)-8-[3-(pyridin-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(azocan-1-yl)-N-[(2R)-1-(benzyloxy)-3-hydroxypropan-2-yl]propanamide
7,7-dimethyl-2-[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-1H-pyrazole-3-carboxamide
1-[9-benzyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-3-(methylsulfanyl)propan-1-one
N-cycloheptyl-3-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]propanamide
ethyl 4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
4-(2-ethoxyphenyl)-3-[(4-hydroxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-2-(5-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}furan-2-yl)-1H-1,3-benzodiazole
(3R,4S)-4-(3-methoxyphenyl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)pyrrolidin-3-amine
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-phenyl-1H-1,2,3-triazole-5-carboxamide
5-methyl-4-[3-(morpholin-4-yl)pyrrolidin-1-yl]thieno[2,3-d]pyrimidine-6-carboxylic acid
2-{5-[(1,1-dioxo-1λ6-thian-4-yl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
1-(2-{1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
7-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
{5-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)methyl]furan-2-yl}methanol
1-cyclopentyl-4-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-1,4-diazepane
6-(3,5-difluorophenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
4-{3-[3-(hydroxymethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-methyl-9-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-phenyl-2,9-diazaspiro[5.5]undecane
1-(cyclohexylmethyl)-N,N-dimethyl-5-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{[4-(4-chloro-2-fluorophenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
1-(1,3-dihydroxypropan-2-yl)-5-oxopyrrolidine-3-carboxylic acid
1-(4-methoxyphenyl)-3-methyl-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-one
1'-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-propoxyethan-1-one
(1R,2R,6S,7S)-N-[4-(1,3-thiazol-4-yl)phenyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}acetamide
7-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-ethyl-8-(furan-3-ylmethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-fluorophenyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)morpholine
3-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-N,N-dimethylpropanamide
9-(2-propoxyacetyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-[1-(propan-2-yl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-{[1-(carbamoylmethyl)piperidin-4-yl]formamido}-2-(4-methylphenyl)acetic acid
5-chloro-6-{3-[(2-fluorophenyl)methoxy]phenyl}-2-methylpyrimidin-4-ol
3-ethyl-1-{4-[ethyl(methyl)amino]pyrimidin-2-yl}piperidin-3-ol
N-[(3-chlorophenyl)methyl]-N-cyclopropyl-1H-1,2,4-triazole-5-carboxamide
4-{1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-3-yl}morpholine
2-amino-4-(3-ethyl-1,2-oxazol-5-yl)-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
(1S,6R)-3-methyl-9-[(2,3,4-trimethoxyphenyl)methyl]-3,9-diazabicyclo[4.2.1]nonane
1-(2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetyl)piperidine-4-carboxamide
6-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-cyclopentanecarbonyl-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-4-carboxamide
2-(2-acetamidoethyl)-N-(4-phenoxyphenyl)piperidine-1-carboxamide