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5-{2-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}pyrrolidin-2-one
4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-methyl-5-propylpyrimidine
4-(2,6-dimethylpyridin-3-yl)-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}pyrimidine
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
(3aS,6aS)-5-[(benzylcarbamoyl)methyl]-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N2,N4,N4,5-tetramethyl-N2-(quinoxalin-2-ylmethyl)pyrimidine-2,4-diamine
6-methyl-8-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene
1-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-5-methyl-1H-1,2,3,4-tetrazole
4-[(1R,9aR)-octahydro-1H-quinolizine-1-carbonyl]-1-phenylpiperazin-2-one
2-[2-(2-fluoro-6-methoxyphenyl)-4-methylphenoxy]acetamide
(1R,5R)-3-(1-benzoxepine-4-carbonyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(pyridin-2-yl)acetamide
8-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-oxa-8-azaspiro[4.5]decane
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-4-hydroxy-3-methylbenzamide
1-(benzenesulfonyl)-N-[2-(2,4-dimethylphenoxy)ethyl]-N-methylcyclopropane-1-carboxamide
3-{[cyclohexyl(pyridin-2-ylmethyl)carbamoyl]amino}-N,4-dimethylbenzamide
ethyl 5-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-pyrazole-4-carboxylate
1-ethyl-4-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]piperazine
3-(4-chloronaphthalen-1-yl)-1-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}urea
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-3-methyl-1H-pyrazole-5-carboxamide
N-(4-{[ethyl(pyridin-4-ylmethyl)carbamoyl]methyl}phenyl)butanamide
ethyl 1-[2-(pyridin-3-yloxy)propyl]-1H-imidazole-2-carboxylate
4-[1-cyclohexyl-5-(2-methanesulfonylethyl)-1H-1,2,4-triazol-3-yl]benzamide
N-(3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-5-methylthiophen-2-yl)-2,2-dimethylpropanamide
(3R,4S)-1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-cyclopropylpyrrolidin-3-amine
5-(5-chlorothiophen-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-methyl-6-(3-methyl-3-phenylpiperidine-1-carbonyl)-4H-pyran-4-one
4-ethyl-5-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
2-ethyl-9-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
N-methyl-4-[(2-methylprop-2-en-1-yl)oxy]-N-[1-(pyridin-2-yl)propan-2-yl]benzamide
(1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperidin-3-yl)methanol
[(2S)-1-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-2-yl]methanol
2-methyl-8-(quinoxaline-6-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
prop-2-en-1-yl 4-[(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carboxylate
4-ethyl-1-methyl-3-[1-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-cyano-N-[(3R,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]pyridine-3-carboxamide
[(4-cyclopropyl-5-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
2-(2H-1,3-benzodioxol-5-yl)-1-[1-(1-methylpiperidin-4-yl)piperidin-4-yl]-5-(trifluoromethyl)-1H-1,3-benzodiazole
4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
1-[4-(oxolan-2-ylmethoxy)phenyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-1,4-diazepan-5-one
(2S,4R)-1-benzyl-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,2-dihydroquinolin-2-one
2-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carbonyl]pyridine
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide