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2,3-dimethyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)quinoxaline-6-carboxamide
3-{1-[(4-chloro-3-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
5-(piperidin-4-yl)-3-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5-propylimidazolidine-2,4-dione
1-[2-(3-fluorophenyl)piperidin-1-yl]-3-methoxypropan-1-one
4-ethyl-5-methyl-N-[3-(oxolan-3-yl)propyl]pyrimidin-2-amine
2-{4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazin-1-yl}benzonitrile
N-(1H-indol-5-yl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine-4-carboxamide
(1S,5R)-3-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)morpholine-2-carboxylic acid
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
N-cyclopropyl-3-[4-({[(5-methyl-1H-imidazol-4-yl)methyl]carbamoyl}amino)phenyl]propanamide
4-{1-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]piperidin-3-yl}benzoic acid
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxane-4-carbonyl)piperidine
1'-[(5-ethylpyridin-2-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(3S)-N-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-amine
N-methyl-N-(pyridin-3-ylmethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-5-phenylpentan-1-one
5-({3-[2-(2H-1,3-benzodioxol-5-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)-N-(propan-2-yl)pyrimidin-2-amine
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2,5-dimethylbenzamide
N3-[(4-chlorophenyl)methyl]-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)methyl]methanesulfonamide
5-[5-(4-fluoro-2-methoxyphenyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
5-chloro-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-3-methyl-N-(oxolan-2-ylmethyl)-1H-indole-2-carboxamide
benzyl 7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxylate
5-ethyl-N,2,3-trimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
6-(pyrrolidin-1-ylmethyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4-oxazepan-6-ol
1-[3-({[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl]amino}methyl)phenyl]ethan-1-one
N-[(4-fluorophenyl)methyl]-3,5-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-(morpholin-3-yl)ethan-1-one
5-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}-8-methylquinoline
2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)pyridine-3-carboxamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-5-methyl-1H-indazole-3-carboxamide
1-methyl-4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidine-1-carboxamide
1,3-dimethyl-5-{octahydropyrrolo[1,2-a]piperazin-2-yl}-1H-pyrazolo[3,4-d][1,3]thiazole
methyl 3-(2-chlorobenzamido)-6-{[4-(hydroxymethyl)piperidin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
(3S,4S)-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
N,N-diethyl-1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
N-methyl-3-[1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidin-3-yl]-N-(1-methylpiperidin-4-yl)propanamide
(4aR,8aS)-1-butyl-6-[(2-methylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
3-(4-fluorophenyl)-6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridazine
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[3-(1H-indazol-1-yl)propyl]acetamide
2-(4-fluorophenyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]morpholine
methyl 6-cyclobutanecarbonyl-2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)propanamide
5-{[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]carbamoyl}thiophene-2-carboxylic acid
[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]diphenylmethanol
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
5-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide