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N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)quinoxalin-2-amine
3-(3-methoxypropyl)-1-[2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]piperidine-3-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}oxolane-2-carboxamide
(4aR,8aR)-2-(5-methyl-1,3-oxazole-4-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-[(3S,4R)-1-(3,6-dimethylpyrazin-2-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole
(2S,4S)-4-amino-N,N-diethyl-1-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]pyrrolidine-2-carboxamide
4-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrimidin-2-amine
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}[(2-fluorophenyl)methyl]amine
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
4-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
2-{1-[1-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
2-[5-(2-methylpyridine-3-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
2-(dimethylamino)-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-(2-oxopyrrolidin-1-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)quinoline-3-carboxamide
(1S,6R)-9-(azepane-1-sulfonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[3-(pyrrolidin-1-yl)propyl]benzamide
{3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
3-(1H-1,3-benzodiazol-2-yl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}propanamide
3-{2-azaspiro[4.4]nonan-2-ylmethyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl){[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}amine
6-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-N,N-dimethylpyrazine-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-butyl-N-(thiophen-3-ylmethyl)acetamide
1-(3-methoxyphenyl)-4-{[4-(methylamino)pyrimidin-2-yl]amino}pyrrolidin-2-one
{1-[(3-methylquinoxalin-2-yl)methyl]-3-(3-phenylpropyl)piperidin-3-yl}methanol
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
(2S,4R)-4-amino-1-(2,6-dimethoxypyridine-3-carbonyl)-N-ethylpyrrolidine-2-carboxamide
8-{[4-(difluoromethoxy)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
N,N-diethyl-1-{1-[(2-methoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
3-benzyl-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazin-2-one
N-(3-ethoxyphenyl)-2-[4-(thiophene-2-carbonyl)morpholin-3-yl]acetamide
9-[1-(4-chlorophenyl)cyclopropanecarbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-{4-[1-(furan-2-ylmethyl)piperidin-4-yl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-{[5-(1-benzylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
2-(5-methyl-1H-pyrazol-1-yl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(quinoline-6-carbonyl)pyrrolidin-3-yl]methanol
3-[5-({cyclopentyl[(3-methylthiophen-2-yl)methyl]amino}methyl)thiophen-2-yl]prop-2-yn-1-ol
3-methyl-3-{[3-(methylsulfanyl)phenyl]methyl}-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
(1S,5R)-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-methyl-3-oxo-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
N-({1-[(2,3,6-trifluorophenyl)methyl]pyrrolidin-3-yl}methyl)butanamide
2-ethyl-1-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidine
1-(but-2-ynoyl)-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
2-(methoxymethyl)-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,3,4-oxadiazole
3-amino-N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)benzamide
N-benzyl-N-ethyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
4-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]thiomorpholine
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(pyrrolidin-1-yl)ethan-1-one