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(2R,3R,6R)-5-cyclopropanecarbonyl-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}phenoxy)acetic acid
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-cyclopropyl-4-hydroxy-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
N-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]-6-methyl-1,4-dihydropyridin-4-one
N-cyclooctyl-2-{[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}acetamide
1-(adamantan-1-yl)-4-(2-methoxypyridine-3-carbonyl)piperazine
N-[2-hydroxy-1-(thian-4-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
2,3-difluoro-6-methoxy-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]benzamide
1-[(3-fluorophenyl)methyl]-4-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-1,4-diazepane
N-[(3S,4R)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-({5-[(2-phenoxyethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)pyridine-2-carboxamide
5-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-1,3-benzodiazole
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-ol
N-(3-phenylprop-2-yn-1-yl)-7-(propan-2-yl)-N-propyl-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
7-(cyclopropylmethyl)-2-(2-hydroxynaphthalene-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-2-(4-hydroxyphenyl)ethan-1-one
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(3,3,3-trifluoropropyl)piperidine
methyl 4-{[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}butanoate
{1-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}methanol
N-(2,2-dimethyloxan-4-yl)-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
7-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[1-(pyridin-2-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
6-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
5-methoxy-2-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1,4-dihydropyridin-4-one
4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
2-{3-oxo-9-[2-(phenylsulfanyl)ethyl]-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
2-(2,6-dimethoxy-4-methylphenyl)-4-(3,3,3-trifluoropropyl)pyrimidine
(2S)-2-hydroxy-2-phenyl-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,2-oxazol-3-yl)methyl]amine
3-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-1-methyl-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
(4S)-3-[(4-methoxypyridin-2-yl)methyl]-4-phenyl-1,3-oxazolidin-2-one
(2S,4S)-4-amino-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-methylpyrrolidine-2-carboxamide
1-(2,3-dihydro-1H-inden-5-yl)-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-(cyclopropylmethyl)-1-(5-methoxypyrimidin-2-yl)piperidine-3-carboxylic acid
N-{2-[3-(morpholin-4-ylmethyl)phenoxy]propyl}propanamide
4-(4-{1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
3-methyl-2-[(1S)-1-(5-methyl-4-phenyl-1H-imidazol-1-yl)ethyl]pyridine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(5-methylfuran-2-yl)pyridine-3-carbonitrile
1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one