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N-[2-(dimethylsulfamoyl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
5-cyclopropanecarbonyl-1'-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-cyclopentyl-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
N,2-dimethyl-7-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[3-(3-methylphenoxymethyl)piperidin-1-yl]propan-1-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
4-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
N-ethyl-2-methyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
1-{4-[2-methoxy-4-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
(2S,4R)-4-amino-1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N,N-diethylpyrrolidine-2-carboxamide
5-methyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1,3-oxazole-4-carboxamide
1-methyl-2-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}azepane
(1S,5R)-N-cyclohexyl-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-benzyl-4-hydroxy-N-(3-hydroxypropyl)-2-(4-methylphenyl)pyrimidine-5-carboxamide
({2-[(2-fluorophenyl)methoxy]-7-methoxyquinolin-3-yl}methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
1-(5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)piperazine
methyl 2-[methyl(2-methylpropyl)sulfamoyl]-6-[(2-methylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-4-oxobutanoic acid
N-tert-butyl-2-methyl-3-[2-(1H-1,2,3,4-tetrazol-5-yl)acetamido]benzamide
N-[2-(pyrrolidin-1-yl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-5-(trifluoromethyl)pyridine
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
5-(1H-indole-2-carbonyl)-1-methyl-N-[3-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-3-yl)pyrrolidin-2-one
N-(3-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}-2,5-dimethyl-1H-pyrrol-1-yl)acetamide
N-[(5-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
2-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-1,2-oxazinane
N-{1-[2-(2-benzyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1H-pyrazol-4-yl}-2-phenoxyacetamide
N-(2-hydroxyethyl)-2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
1-(2-{4-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
N-methyl-4-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyridin-2-amine
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}urea
2-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}methyl)benzonitrile
4-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-[2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole
3-hydroxy-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)benzamide
1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N,N-dimethyl-1-(2-methylpropyl)-5-{[2-(thiophen-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[4-({4-[2-(methylsulfanyl)pyridine-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-ol
N-{5-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazol-7-yl}acetamide
4-ethyl-3-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-N-(propan-2-yl)-1-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]pyrrolidine-2-carboxamide
2-[4-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]acetic acid
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperazine
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}cyclopropanamine
1-cyclopentyl-N-(3-methylbutyl)-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}-4-phenylpyrrolidin-2-one
7-{2-methylthieno[3,2-d]pyrimidin-4-yl}-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine