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(2S,4S)-4-amino-1-{[(1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl]methanesulfonyl}-N-ethylpyrrolidine-2-carboxamide
1-[2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]-3,3-dimethylurea
5-{[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
3-cyclobutyl-4-(4-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-methyl-2-{[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}pyrimidin-5-yl)ethan-1-one
(1R,7S)-6-(3-phenoxyazetidine-1-carbonyl)-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidine
7-fluoro-4-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}quinazoline
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]propanamide
methyl 4-(methylsulfanyl)-2-[2-(2,3,6-trimethylphenoxy)acetamido]butanoate
5-[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
2-(3-{1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-6-methylpyridine
3,6-dimethyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-benzofuran-2-carboxamide
2-(2,4-dimethoxyphenyl)-3-methoxypyridin-4-amine
N-(cyclohex-1-en-1-ylmethyl)-3-(1-methylpiperidin-2-yl)propanamide
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(piperidin-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(1H-pyrazol-1-yl)benzamide
N,N-dimethyl-5-{[(4-methylphenyl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-chloro-6-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]pyridine-2-carboxylic acid
methyl[(2-methyl-1,3-oxazol-4-yl)methyl](quinolin-2-ylmethyl)amine
3-{5-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-butyl-4-ethyl-1-[2-oxo-2-(2-phenylmorpholin-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyrimidin-2-amine
1-(4-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
3-(5-chloro-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-methyl-1H-pyrazol-3-yl)-5-methyl-1,2-oxazole
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-[2-(pyrazin-2-yl)ethyl]acetamide
1-benzoyl-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}piperidine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[N-benzyl-1-(1-methyl-5-phenyl-1H-pyrrol-2-yl)formamido]propanamide
5-methyl-5-phenyl-1-{3-[(pyridin-3-yl)amino]propyl}piperidin-2-one
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-4-ylmethyl)piperidine
2-(4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenoxymethyl)pyridine
1-(4-methylphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidin-4-amine
2-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
1-(1H-imidazol-2-ylmethyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
7-(cyclopropylmethyl)-N-(2-hydroxyethyl)-N-methyl-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-1H-1,3-benzodiazole
(2S,4R)-N,N-diethyl-1-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]pyrrolidine-2-carboxamide
N,N-diethyl-2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoacetamide
(2S,4S)-4-amino-N-ethyl-1-(4-methoxybenzenesulfonyl)pyrrolidine-2-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(2H-1,3-benzodioxol-5-yl)-3-phenylpropanamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
4-[ethyl({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl})amino]butan-1-ol
(1R,7S)-3-(4-fluoro-2-methylphenyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(3-hydroxypropyl)-1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(morpholin-4-yl)acetamide