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3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidine
3-(propan-2-yl)-5-{1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]pyrrolidin-2-yl}-1,2,4-oxadiazole
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-chloro-4-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
4-(2-amino-5-ethylpyrimidin-4-yl)-1-(3,5-dimethylphenyl)piperazin-2-one
4-[2-(4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H-1,2,3-triazol-1-yl)ethyl]-1,3-thiazol-2-amine
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-2-carboxamide
methyl[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl][1-(pyridin-4-yl)ethyl]amine
{4-[(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl)methyl]phenyl}methanol
2-[4-(9H-purin-6-yl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
4-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-(trifluoromethyl)pyrimidine
5-(4-ethylpiperazin-1-yl)-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2,3-dihydro-1-benzofuran-2-carboxamide
5-(3-methoxyphenoxymethyl)-N-(piperidin-3-yl)-1H-pyrazole-3-carboxamide
methyl 2-({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
2-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-imidazol-2-yl}pyridine
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
1-cyclohexyl-4-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperazine
2-{1-[(1-methyl-1H-imidazol-2-yl)methyl]azetidin-3-yl}pyridine
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-ol
9-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-methyl-2-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}pyridine
3-[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
4-hydroxy-1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperidine-4-carboxylic acid
2-(7-chloro-4-methylquinolin-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-{4-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
3-hydroxy-3-({methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
1-cyclopentyl-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(1H-indol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(2-methyl-1,3-thiazol-4-yl)methyl][4-(1H-pyrazol-1-yl)butan-2-yl]amine
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)cyclopropanecarboxamide
1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-methyl-1-[1-(1,2-oxazol-3-yl)ethyl]urea
N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-1,3-oxazole-4-carboxamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N-[1-(3,5-difluorophenyl)cyclopropyl]-3-(2-oxopiperidin-1-yl)propanamide
2-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-3-(trifluoromethyl)pyridine
4-ethyl-3-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
1-[(2,6-difluorophenyl)methyl]-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-chloro-N-(1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-(3-chlorophenyl)-3-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]urea
2-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-2-yl}pyridine
1'-(2,3-dihydro-1H-indene-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-ethyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide