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5-(1-{[5-(2-chlorophenyl)furan-2-yl]methyl}pyrrolidin-2-yl)-3-methyl-1,2-oxazole
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrazole-3-carbonyl)piperidine
N-ethyl-N-[(1-methylpyrrolidin-3-yl)methyl]-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
(3S,4R)-4-methyl-1-[3-(1H-pyrazol-4-yl)benzoyl]piperidine-3,4-diol
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}urea
1-(2-hydroxyethyl)-4-(1-phenylpiperidin-4-yl)-1,4-diazepan-6-ol
3-{[(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amino]methyl}-1-methyl-1,2-dihydroquinolin-2-one
7-(furan-3-ylmethyl)-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-(1H-imidazol-4-ylmethyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
1-cyclobutanecarbonyl-N-(1-phenylpiperidin-4-yl)piperidine-4-carboxamide
2-benzyl-8-[2-(2-methylphenyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
9-[(3,4-difluorophenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R,6R)-11-methoxy-4-(1-methylpiperidine-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(4-chloro-2-methylbenzoyl)-2-(3-methoxypropyl)piperidine
4-(2-methylphenoxy)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
3-[(3R,4S)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(2S,4R)-4-amino-1-(6-aminopyridine-3-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(1H-indol-3-yl)acetamide
3-[({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-N-methylbenzamide
ethyl 4-({1-[4-(2H-1,3-benzodioxole-5-amido)phenyl]piperidin-4-yl}amino)piperidine-1-carboxylate
N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}-2-(pyrrolidin-1-yl)benzamide
2-(5-acetylthiophen-3-yl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]acetamide
1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(3R,9aR)-8-(3,5-difluorobenzoyl)-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
N-methyl-2-(1-methyl-1H-imidazol-2-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]({[7-chloro-2-(2,3-dimethoxyphenyl)quinolin-3-yl]methyl})amine
1-{3-oxo-3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]propyl}-1,2-dihydropyridin-2-one
6-methyl-4-[4-(pyridin-3-yl)piperazin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
2-[2-({[2-(3,5-dimethylphenoxy)ethyl](methyl)carbamoyl}amino)phenyl]-N,N-dimethylacetamide
3-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1-[3-(pyridin-3-yl)propyl]urea
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(methylsulfamoyl)ethyl]acetamide
5-[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-(3-ethylphenyl)-3-{[(2S)-1-methoxypropan-2-yl]amino}propanamide
[(2S,6S)-11-methoxy-4-(2,2,6,6-tetramethylpiperidin-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-(5-fluoro-2-methoxyphenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
ethyl 4-(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazole-4-amido)piperidine-1-carboxylate
3-methyl-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3-phenylpiperidine
7-[3-(1,3-benzothiazol-2-yl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-2-phenyl-2,3-dihydro-1H-indene-1,3-dione
1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
1-(oxolane-3-carbonyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
2-methyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzoyl]piperidine
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(quinolin-6-yl)pyridine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(5-methoxy-1H-indol-2-yl)methyl]propanamide
methyl 3-{6-[(3-methoxyphenyl)methoxy]-2-oxo-4-(2-phenoxypropanoyl)-1,4-diazepan-1-yl}propanoate
2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one