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2-methyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(oxan-4-yl)piperidine-3-carboxamide
N-cyclopropyl-5-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}thiophene-2-carboxamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(2,2,2-trifluoroethyl)propanamide
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}thian-4-amine
N-[2-(1H-imidazol-4-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-(propan-2-yl)-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-5-[(2,2,2-trifluoro-1-phenylethoxy)methyl]-1H-1,2,4-triazole
(4aR,7aS)-N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl][(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
N-(1-methanesulfonylpiperidin-4-yl)-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-{1-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
2-(4-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
methyl 3-{4-[2-amino-3-cyano-6-(3-methylphenyl)pyridin-4-yl]-1H-pyrazol-1-yl}propanoate
1-ethyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
1-[3-(2-{[(cyclopropylmethyl)(propyl)amino]methyl}-4-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
N'-[(6-chloropyridin-3-yl)methyl]-N-cyclopentylbutanediamide
2-(1-benzylpiperazin-2-yl)ethan-1-ol
2-{1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-5-fluoro-1H-1,3-benzodiazole
1-[(1-methyl-1H-indol-3-yl)methyl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
10-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octane-8-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
({3-[(dimethylamino)methyl]-4-methoxyphenyl}methyl)(methyl)[(2-methylpyridin-4-yl)methyl]amine
(4aS,8aR)-6-(dimethyl-1,3-oxazole-4-carbonyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
1-[(3-methylphenyl)methyl]-3-{[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methyl}urea
(1R,5S)-6-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-6-azabicyclo[3.2.1]octane
N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
1-(cyclohexylmethyl)-5-{[(1-hydroxycyclohexyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl({[1-(propan-2-yl)-1H-imidazol-5-yl]methyl})[2-(pyridin-2-yl)ethyl]amine
1-(2-methylphenyl)-3-[1-(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2,6,8-trimethylquinoline-4-carboxamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
(2S,4S)-4-amino-1-[(3-chloro-4-ethoxyphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
4-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridine-6-carboxamide
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
4-[1-(tert-butylcarbamoyl)piperidin-3-yl]benzoic acid
1-[3-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
N-(2-acetamidoethyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-(2-chlorophenyl)-3-{1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
1-(cyclohexylmethyl)-N-cyclopropyl-5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazole
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl})amine
3-({[2-(quinolin-8-yloxy)ethyl]amino}methyl)piperidin-3-ol
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-4-ol
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(oxolan-3-ylmethyl)piperazine
1-(morpholin-4-yl)-3-[1-(oxolan-3-ylmethyl)piperidin-4-yl]propan-1-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide