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[3-(cyclopropylmethyl)-1-(4-fluoro-3-methylbenzoyl)piperidin-3-yl]methanol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
1-[1-(1-benzyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-4-phenylpiperazine
1-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]azepan-2-one
(1S,6R)-9-[4-(4-chlorophenyl)butanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[4-(furan-3-carbonyl)piperazin-1-yl]-4-methyl-6-(trifluoromethyl)pyrimidine
6-(3-fluoro-4-methoxyphenyl)-N-(2-methoxyethyl)-N-(propan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(9H-purin-6-yl)piperazin-2-yl}ethan-1-ol
3-chloro-5-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(cyclohexylmethyl)-5-(cyclopropylamino)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]methyl}benzoic acid
5-{[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]methyl}-3-(propan-2-yl)-1,2,4-oxadiazole
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
N-{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}-N-(3-methoxypropyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
3-(2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-(phenoxymethyl)-1H-1,3-benzodiazole
4-({[2-amino-6-(propan-2-yl)pyrimidin-4-yl]amino}methyl)-1-phenylpyrrolidin-2-one
8-[(2,2-dimethyloxan-4-yl)methyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(4-chlorophenyl)-N,N-dimethyl-3-phenylpropanamide
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-(morpholin-4-yl)butan-1-one
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-(1H-pyrazol-1-yl)butan-1-one
4-{1-cyclohexyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}benzonitrile
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N,N-dimethyl-3-(2-{[({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)carbamoyl]amino}phenyl)propanamide
N-(1H-1,2,4-triazol-3-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-butyl-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperazin-2-one
5-butyl-1'-(1-ethyl-1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{4-[(oxan-4-ylmethyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-[5-({[2-(dimethylamino)ethyl][(3-methylthiophen-2-yl)methyl]amino}methyl)thiophen-2-yl]prop-2-yn-1-ol
2-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-5-methylphenol
(1S,6R)-N-(3-benzylphenyl)-3-methyl-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N6-benzyl-N5-methyl-N5-(oxan-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]acetamide
3-({[(5-tert-butyl-2-methoxyphenyl)carbamoyl]amino}methyl)-N,N-dimethylbenzamide
1-ethyl-N-(3-phenylpropyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(azocan-1-yl)-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
(2R,3R,6R)-3-phenyl-5-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,5R)-3-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(carbamoylmethyl)-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
6-fluoro-2-({[(1s,4s)-4-aminocyclohexyl]amino}methyl)quinolin-4-ol
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
2-methoxy-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
2-[6-(2-ethylpiperidin-1-yl)-2-methylpyrimidin-4-yl]ethan-1-amine
1-ethyl-N-(2-ethyl-2,5-dihydroxypentyl)-2-oxo-1,2-dihydropyridine-4-carboxamide
1-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepan-6-ol
4-{[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)amino]methyl}-2,6-dimethylphenyl acetate
2-(dimethylamino)-7-[2-(1H-imidazol-2-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one