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N-[(5-{[3-(2-aminoethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
[1-(4-ethoxypyrimidin-2-yl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
6-(benzyloxy)-1-cyclohexyl-4-(pyridin-4-ylmethyl)-1,4-diazepan-2-one
N-(4-acetylphenyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[2-(pyrrolidin-1-yl)ethyl]piperidine
N-ethyl-5-{4-[2-(pyrrolidin-1-yl)ethyl]piperazine-1-carbonyl}pyrimidin-2-amine
1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}pentan-1-one
(2S,4S)-4-amino-1-(2-amino-1,3-benzothiazole-5-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-cyclohexyl-4-[2-(trimethyl-1H-pyrazol-1-yl)acetamido]piperidine-1-carboxamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-[(naphthalen-1-ylmethyl)amino]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperazin-2-one
(1S,4S)-2-(3,4-difluorophenyl)-5-[2-(trifluoromethyl)benzoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-(2-chlorophenyl)-4-[(2,6-difluoro-3-methylphenyl)methyl]piperazin-2-one
2-ethyl-4-methyl-3-oxo-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine-1-carboxamide
N-(furan-3-ylmethyl)-N,7-dimethyl-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N,5-diethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
2-(4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
methyl 3-(acetamidomethyl)-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
(1S,5R)-6-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
3-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-1-(5-fluoropyridin-3-yl)urea
4-(4-ethyl-1H-pyrazol-5-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine
N-cyclopentyl-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
2-(4-chlorophenyl)-4-{2-methylpyrido[2,3-d]pyrimidin-4-yl}morpholine
N-{[4-(1H-imidazol-1-yl)phenyl]methyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-[(3S,5S)-5-[(furan-3-ylmethyl)(methyl)carbamoyl]-1-methylpyrrolidin-3-yl]morpholine-4-carboxamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
1,3-dimethyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(2,3-difluorophenyl)-1-(3-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
1-{2-[(4-chlorophenyl)methoxy]ethyl}-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
4-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-6-hydroxy-N,N-dimethyl-1,4-diazepane-1-carboxamide
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)(pyrazin-2-ylmethyl)amine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-[(naphthalen-1-ylmethyl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2-oxoazonan-1-yl)acetamide
2-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(furan-2-ylmethyl)(3-methylbutan-2-yl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-(3-phenylpropyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
(3S,5R)-1-[2-(2-methoxyphenyl)acetyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
2-chloro-4-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}phenol
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
3-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]morpholine-2-carboxylic acid
8-methyl-2-propyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[(3S,4S)-3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-4-hydroxypyrrolidin-1-yl]-2-methoxyethan-1-one
N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)(pyridin-4-ylmethyl)amine
4-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}phenyl)-2-methylbut-3-yn-2-ol