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4-(3-acetylphenyl)-3-[(4-hydroxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(1H-1,2,4-triazole-5-carbonyl)piperidine
N3-butyl-N3-methyl-N5-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-ethyl-N-[2-(ethylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
2,3-dimethyl-7-[3-(2-methyl-1H-imidazol-1-yl)butanoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
2-(dimethylamino)-7-(quinoxaline-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[(3R,4S)-1-[(2-methyl-1-benzothiophen-3-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-(cyclobutylmethyl)-3-hydroxy-3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}piperidin-2-one
2-benzyl-9-[(2E)-2-methylbut-2-en-1-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3-chloro-4-fluorophenoxy)-1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
methyl[(4-methyl-1H-imidazol-5-yl)methyl][3-(1-methyl-1H-pyrazol-4-yl)propyl]amine
3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-1-[2-(4-sulfamoylphenyl)ethyl]urea
1-(1-methyl-1H-pyrazole-4-carbonyl)-4-(pyrrolidine-1-carbonyl)piperidine
4-(4-phenyl-1H-1,2,3-triazol-1-yl)-1-(1,3-thiazol-2-ylmethyl)piperidine
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-4-(4-chlorophenyl)butanamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
2-{2,7-diazaspiro[4.5]decane-7-carbonyl}-6-methoxyphenol
(4aS,8aR)-1-(3-methoxypropyl)-6-(3-phenylpropanoyl)-decahydro-1,6-naphthyridin-2-one
2-(2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)pyridine
N-{[5-(6-phenylpyridazin-3-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-{[1-(3,5-dimethylfuran-2-carbonyl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
1-(6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-2-yl)ethan-1-ol
N-[2-(1,3-benzoxazol-2-yl)ethyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(1H-1,2,4-triazol-1-yl)butanamide
2-methyl-4-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}phenol
(1R,2R)-N-methyl-2-phenyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}cyclopropane-1-carboxamide
N-[(3R,4R)-1-(3-fluoropyridin-2-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
N-(3-hydroxypropyl)-N-methyl-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-(4-{[ethyl(oxan-4-ylmethyl)amino]methyl}phenyl)ethan-1-one
5-(3-methylphenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-2-(2,5-dimethoxyphenyl)ethan-1-one
N-(1-{7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
5-(propan-2-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]thiophene-3-carboxamide
methyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
(1S,5R)-3-[2-(4-fluorophenoxy)ethyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4R)-1-(3-fluoropyridin-4-yl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-[(2-chlorophenyl)methyl]-3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]propanamide
4-(4-fluorophenyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-4-oxobutanamide
(3aS,6aS)-2-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-cyclopentyl-4-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]piperazin-2-one
N-[(3S,4R)-1-(5-hydroxypyrazine-2-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
2-benzyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1,3-thiazole-4-carboxamide
3-(3-methoxyphenyl)-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-pyrazole-4-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
3-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-N,N-dimethylpyrazin-2-amine
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1,3-thiazol-4-ylmethyl)piperidine
2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}-N,N-dimethylacetamide