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3-[({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]-2,2-dimethylpropan-1-ol
1-(3,5-dimethylphenyl)-N-[(4-fluoro-3-methoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[(5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}thiophen-2-yl)methyl]pyrrolidine
6-cyano-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyridine-3-carboxamide
2-(2,4-dichlorophenoxy)-1-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]ethan-1-one
5-(1H-pyrazol-3-yl)-2-(pyridin-3-yl)-1,3-benzoxazole
(2S,4S)-4-amino-N,N-diethyl-1-(2,6,8-trimethylquinoline-4-carbonyl)pyrrolidine-2-carboxamide
N-(2-methyl-1-benzofuran-5-yl)-2-propyl-2,5-dihydro-1H-pyrrole-1-carboxamide
N-(3-fluoro-4-methylphenyl)-4-[(1-methylpiperidin-4-yl)methyl]piperazine-1-carboxamide
N-{1-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methylthiophene-3-carboxamide
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
1-[3-(diethylamino)pyrrolidin-1-yl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
8-(8-chloroquinoline-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(dimethylamino)-N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]-2-(3-methylphenyl)acetamide
N-butyl-N-cycloheptyl-5-[(dimethylamino)methyl]furan-2-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
N-ethyl-5-{1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-4-methyl-1,3-thiazol-2-amine
propan-2-yl 2-chloro-5-[2-(1H-1,2,4-triazol-5-yl)benzamido]benzoate
6-chloro-N,N-dimethyl-3-({[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
3-cyclopentyl-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]propan-1-one
7-(2-cyclohexylethyl)-2-(2-methylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(pyrrolidine-1-carbonyl)-5-{[(thiophen-3-ylmethyl)amino]methyl}phenyl]pyridine-2-carboxamide
N,1-dimethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(pyridin-3-yl)propanamide
5-benzyl-4-(2,2-dimethylpropanoyl)-1-(3-methoxyphenyl)piperazin-2-one
3-benzyl-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
7-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-indole
2-hydroxy-N-[2-(4-methylpiperazin-1-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]acetamide
N-methyl-2-[4-({[1-(5-methylpyridin-2-yl)propyl]carbamoyl}amino)phenyl]acetamide
5-{[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
5-{[1-cyclohexyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
4-(2H-1,3-benzodioxol-5-yl)-3-(morpholin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(1-butyl-3-methyl-1H-1,2,4-triazol-5-yl)-2-methyl-1H-1,3-benzodiazole
5-[3-(3-methoxybenzoyl)piperidine-1-carbonyl]-2-methylpyridine
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-4-(trifluoromethyl)benzene-1-sulfonamide
1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-4-phenoxybutan-1-one
1-[(3-methylphenyl)methyl]-4-[2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
5-methyl-2-(3-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N-[2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)quinolin-6-yl]acetamide
2-{[2-(1,1-dioxo-1λ6-thiomorpholine-4-carbonyl)phenyl]amino}acetic acid
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-[(4-methylpiperidin-1-yl)methyl]furan-2-carboxamide
1-[(3-fluorophenyl)methyl]-4-(6-methyl-2-phenylpyrimidin-4-yl)piperazin-2-one
3-(4-chlorophenyl)-N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenylpropanamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-(pyridin-3-yl)acetamide
2-{1-[(3-methylquinoxalin-2-yl)methyl]pyrrolidin-3-yl}benzoic acid
3-cyclohexyl-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
1-[(3,3-dimethylbutan-2-yl)amino]-3-(2,4-dimethylphenoxy)propan-2-ol
1-[2-(4-chloro-2-methylphenoxy)propanoyl]-4-propyl-1,4-diazepan-5-one
1-{3,9-diazaspiro[5.5]undecan-3-yl}-6-methoxyhexan-1-one