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N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(2-methyl-1H-imidazol-1-yl)propanamide
(2S,4S)-4-{[(2,5-difluorophenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
12-(6-hydroxy-1,4-oxazepane-4-carbonyl)-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
(1S,4S)-2-benzyl-5-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-2,5-diazabicyclo[2.2.1]heptane
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1H-pyrazole-3-carboxamide
8-[(3-methylpyridin-4-yl)methyl]-8-azaspiro[4.5]decane-7,9-dione
2-(methylsulfanyl)-3-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(1H-indol-3-yl)-1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
3-chloro-N-cyclopentyl-4-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
5-benzyl-4-ethyl-1-(3-methoxyphenyl)piperazin-2-one
(3R,7S,8aS)-7-{[(2-fluorophenyl)methyl]amino}-3-[(1S)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-[(1S,6R)-6-carbamoylcyclohex-3-en-1-yl]-3,5-dimethyladamantane-1-carboxamide
2-(benzyloxy)-N-{[(2S,4S)-4-fluoro-1-(1-methyl-1H-imidazole-2-carbonyl)pyrrolidin-2-yl]methyl}acetamide
6-[(diethylamino)methyl]-N-(6-methylpyridin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2-methylphenoxy)acetamide
5-chloro-2-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenol
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-imidazole-2-carboxamide
(3aR,6aR)-2-cyclopentyl-N-(2-methanesulfonamidoethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(2R)-1-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]-2-methylpiperazine
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-4-methylpentane-1,2-dione
6-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(1H-1,2,4-triazol-1-yl)benzamide
7-[(2R)-oxolane-2-carbonyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-{3-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]propyl}piperidine-3-carboxamide
4-(2-ethoxyphenyl)isoquinoline
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-3-(piperidin-3-yl)benzamide
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxyethan-1-one
1-(5-ethyl-1,3-oxazole-4-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
8-(1-benzoxepine-4-carbonyl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}cyclopentanamine
ethyl 1-(2,3-dihydro-1H-inden-2-yl)-3-(2-methoxyethyl)piperidine-3-carboxylate
5-{3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-sulfonyl]-4-methylphenyl}-2-methyl-1,3-oxazole
1-(2-methoxyethyl)-6-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
2-cyclopropyl-N-[(2-methoxynaphthalen-1-yl)methyl]pyrimidine-5-carboxamide
(1R,5R)-3-cyclobutanecarbonyl-6-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxylic acid
[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
1-[1-(1-methylcyclopropyl)propan-2-yl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(1S,5R)-6-(2-methoxyethyl)-3-(2-propyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,8aR)-1-butyl-6-[2-(methylamino)-1,3-thiazole-4-carbonyl]-decahydro-1,6-naphthyridin-2-one
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(pyrrolidin-1-yl)butanamide
2,6-dimethyl-4-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)phenyl acetate
2-methyl-6-(4-phenyl-1-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}-1H-imidazol-5-yl)pyridine
4-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-2-propylpyridine
6-[({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amino]pyrazine-2-carboxamide
9-[(4-fluorophenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-({3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)quinoline