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5-{2-[3-(dimethylamino)pyrrolidin-1-yl]-4-(4-methylphenyl)pyrimidin-5-yl}pyridin-2-amine
(4aS,8aS)-2-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-decahydro-2,7-naphthyridin-4a-ol
3-(4-methyl-1,3-thiazol-5-yl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}propanamide
methyl 3-ethyl-2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3H-imidazo[4,5-b]pyridine-6-carboxylate
3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-6-methylpyridin-2-ol
3-{[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}pyridin-1-ium-1-olate
2-(1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidine-3-carbonyl)pyridine
5-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
(4aS,7aR)-1-[(5-fluoro-2-methoxyphenyl)methyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 4-{4-[5-(2-methoxy-2-phenylacetamido)-1H-pyrazol-1-yl]piperidin-1-yl}-4-oxobutanoate
2-(5-methyl-1,2-oxazole-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-hydroxypiperidine-4-carboxylic acid
methyl 3-[(3S,4R)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
5-chloro-2-methoxy-4-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
1-(1-methyl-1H-pyrazole-5-carbonyl)-3-(2-phenylethyl)piperidine
methyl 1-{3-[3-({[(4-fluorophenyl)methyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
2-{4-[1-(pyrimidin-2-yl)piperidin-4-yl]piperazin-1-yl}ethan-1-ol
1-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-(furan-2-yl)ethane-1,2-dione
N,2-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)pyrazine-2-carboxamide
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}acetamide
3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-4-(pyridin-2-ylmethyl)piperazin-2-one
(3R,5S)-N-butyl-5-(3-fluorophenoxymethyl)-1-(2-methylpropyl)piperidine-3-carboxamide
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
methyl (2S,4R)-4-(dimethylamino)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidine-2-carboxylate
8-chloro-2-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}quinolin-4-ol
3-[1-(5-chlorothiophene-2-carbonyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
4-(4-fluorophenoxy)-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidine
2-{2-[(cyclohexylmethyl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
3-[(3R,4S)-1-[(4-fluoro-2-methylphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
methyl 4-[5-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
5-[5-(methoxymethyl)furan-2-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
(2S,4R)-4-[(cyclohexylmethyl)amino]-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[(thiophen-2-ylmethyl)carbamoyl]piperidine-4-carboxylic acid
2-hydroxy-4-(methylsulfanyl)-1-(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)butan-1-one
2-(dimethylamino)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2,3-dihydro-1H-indene-2-carboxamide
4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]-1-{[1,2,4]triazolo[3,4-a]phthalazin-6-yl}piperidine
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(2-phenylethyl)piperidine
1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(1-propyl-1H-1,2,3-triazol-4-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide
1-(adamantan-1-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}urea
6-methyl-N-(2-methylpropyl)-2-oxo-N-(thiophen-3-ylmethyl)-1,2-dihydroquinoline-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-ethyl-N-methylpyrimidine-5-carboxamide
(4aS,8aR)-6-(5-fluoropyrimidin-2-yl)-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
2-amino-3-ethyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[(2-amino-6-methylpyrimidin-4-yl)amino]-N-methyl-2-phenylacetamide
(4-{[(1H-indol-5-ylmethyl)(methyl)amino]methyl}oxan-4-yl)methanol
2-[2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one