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1-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}azepane
3-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-[2-methoxy-4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-{2-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]phenoxy}ethan-1-ol
3-fluoro-N-{[7-(oxan-4-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
3-{[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}phenol
5-fluoro-N2,N4,N4-trimethyl-N2-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-2,4-diamine
3-(4-fluorophenyl)-N-[3-(4-methylpiperazin-1-yl)propyl]-3-phenylpropanamide
4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-propylpyrimidine
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-(2-ethyl-1H-imidazol-1-yl)-N-methyl-N-(pyridin-3-ylmethyl)propanamide
1-(2,6-dimethoxybenzoyl)-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-3-(2-oxoazepan-1-yl)propanamide
3-(1-methylpiperidin-2-yl)-1-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propan-1-one
phenyl (7S,9aR)-7-(cyclohexylmethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
(1S,5R)-6-(4-chloro-3-fluorobenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(4-fluorophenyl)methyl]-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
2-{3-[4-(benzyloxy)piperidine-1-carbonyl]piperidin-1-yl}-6-ethoxy-4-methylquinazoline
N-(2-hydroxyethyl)-5-{1-[2-(pyridin-2-ylsulfanyl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
6-phenyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N,N-dimethyl-4-[({2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)methyl]benzene-1-sulfonamide
2-(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
(3S,4R)-1-[(5-ethylfuran-2-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
N-cyclopropyl-1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-methyl-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}-1H-pyrazole-5-carboxamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
(2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
N-ethyl-2-[4-(8-fluoro-4-oxo-1,4-dihydroquinoline-2-carbonyl)piperazin-1-yl]acetamide
(5S,9aS,9bS)-5-(1-ethyl-1H-imidazol-2-yl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-methyl-1-[1-(pyridin-3-yl)ethyl]urea
2-amino-6-(3-hydroxyphenyl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
2-{2-oxo-2-[3-(propoxymethyl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,2-benzothiazol-3-one
(2E)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
4-[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-1-(1,4-dioxan-2-ylmethyl)-1H-1,2,3-triazole
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
4-ethyl-3-[1-(2-propylpyridine-4-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1,3-benzothiazol-2-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]piperidin-4-amine
3-[(3R,4S)-4-(dimethylamino)-1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-3-yl]propan-1-ol
3-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}imidazolidine-2,4-dione
2-hydroxy-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]pyridine-3-carboxamide
4-[(3S)-3-acetamidopyrrolidin-1-yl]-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
1-(pyridin-3-ylmethyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepane
N,3,6-trimethyl-2-(1H-pyrazol-4-yl)-N-[3-(pyrrolidin-1-yl)propyl]quinoline-4-carboxamide
3-(2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(2-phenylethyl)propanamide
5-chloro-2-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}pyridine
(1R,9S)-5-amino-3-{3-[(dimethylamino)methyl]phenyl}-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-[(1-propyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-inden-2-amine