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1-cyclopentanecarbonyl-4-(3-phenoxyazetidine-1-carbonyl)piperidine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-oxo-2-phenylacetamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}ethan-1-one
1-(5-chloro-2-methoxyphenyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
3-[4-(4-chlorophenoxy)piperidine-1-carbonyl]pyridin-2-ol
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
4-(2,3-dihydro-1H-inden-2-yl)-3-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]piperazin-2-one
5-phenyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,2-oxazole-3-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}ethan-1-one
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
dimethyl({5-[1-(1-methylpiperidin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)amine
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(1-methylpiperidine-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-hydroxyethyl)-6-{6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
5-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-N-(1H-indazol-5-yl)thiophene-2-carboxamide
N-methyl-1-[1-(propan-2-yl)piperidin-4-yl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
3-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
4-(1-{1-[(1-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}ethyl)morpholine
N-{4-[2-(2-ethylpyrimidin-5-yl)-1H-imidazol-1-yl]-2-methylphenyl}butanamide
4-[1-(4-methylquinolin-2-yl)pyrrolidin-3-yl]benzoic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(diethylamino)acetamide
1-(2-amino-5-butyl-6-methylpyrimidin-4-yl)-N-methylpyrrolidine-3-carboxamide
3-[(2-{1-[4-(propan-2-yl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
1-(3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[2,5-difluoro-4-(trifluoromethyl)phenyl]-3-[(3-methyloxetan-3-yl)methyl]urea
1-(oxan-4-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-3-carboxamide
N-[2-(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]pyridine-3-carboxamide
4-({1-[3-(difluoromethoxy)benzoyl]piperidin-2-yl}methyl)morpholine
4-[3-(4-fluorophenyl)propanoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
ethyl 3-{[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]amino}propanoate
(1R,5R)-N-(3,4-dimethylphenyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-cyclobutanecarbonyl-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(2-methoxypyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3-{2-[1-(3-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-3-yl}benzoic acid
(1S,5R)-6-methyl-3-(2-methyl-5-propylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-6-(2-methoxyphenyl)pyridazin-3-amine
4-(2-ethoxyphenyl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}cyclohexanecarboxamide
1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1-[3-(1,3-oxazol-5-yl)phenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
4-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}thiomorpholine
1-[1-(2,4-dimethoxybenzenesulfonyl)piperidin-3-yl]pyrrolidin-2-one
1-{2-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
7-(2-amino-1,3-benzothiazole-5-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(5-chloropyridin-2-yl)-3-(2-phenoxyethyl)piperidine-3-carboxylic acid
1-(4-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-({[2-ethyl-7-(2-hydroxyacetyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)ethan-1-one
1-[3-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)phenyl]ethan-1-one