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1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
5-[4-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-[2-(3,5-dimethylphenoxy)ethyl]-N-methylpropanamide
3-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
4-{1-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}-2-methyl-1,3-thiazole
1'-(pyrazine-2-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(4aS,7aR)-1-(3,5-difluoropyridine-2-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3,3-dimethyl-4-phenyl-1-(pyrrolidine-1-sulfonyl)pyrrolidine
4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
6-(1H-indol-4-yl)-N-(propan-2-yl)pyrimidin-4-amine
N'1-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclopropane-1,1-dicarboxamide
1-methyl-4-phenyl-3-[1-(pyrimidine-4-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(azocan-1-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
1-[4-(propan-2-yl)benzoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
({4-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-yl}methyl)dimethylamine
1-cyclopropanecarbonyl-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
(3S,4S)-4-cyclopropyl-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxylic acid
3-(3-hydroxy-3-methylbutyl)-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}benzamide
2-(4-fluorophenyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}imidazo[1,2-a]pyridine-6-carboxamide
methyl 4-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1H-pyrazole-3-carboxylate
2-(4-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}piperazin-1-yl)-5-fluoropyrimidine
8-methyl-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(3-methoxybenzoyl)-4-(4-methyl-1,3-thiazole-5-carbonyl)piperazine
N-cyclopentyl-4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine
2-{[4-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-propyl-1H-imidazole
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-benzyl-5-(1H-pyrazol-3-yl)furan-2-carboxamide
1-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-1,4-diazepan-6-ol
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
ethyl 2-{[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}acetate
5-{7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane-3-carbonyl}-4-methylpyrimidin-2-amine
1-({1-[(E)-2-phenylethenesulfonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
1-[(3-fluorophenyl)methyl]-4-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)pyrrolidin-2-one
1-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-3-(3-fluorophenyl)propan-1-one
(2S,4R)-1-(2,2-diphenylethyl)-N-methyl-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
(3aR,6aR)-2-(2-aminopyrimidin-4-yl)-5-cyclohexyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-2,3,4-trimethoxybenzamide
6-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-3-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-ethyl-N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-1H-pyrazole-4-sulfonamide
N,1,6-trimethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-[(3-chlorophenyl)methyl]pyrrolidine-2-carboxamide
N-ethyl-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]piperidin-4-amine
4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[1-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)ethyl]morpholine
N-[(4,6-dimethylpyridin-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
methyl 4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine-1-carboxylate
5-fluoro-4-methoxy-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidin-2-amine