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methyl 1-({4-[2-(morpholin-4-yl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
N-[2-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)quinolin-6-yl]acetamide
N-[2-(pyridin-3-yl)ethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
2-cyclopentyl-9-[(3-fluorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
5-[1-(2-methylfuran-3-carbonyl)pyrrolidin-2-yl]-N-(4-methylphenyl)thiophene-2-carboxamide
1-(cyclohexylmethyl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N'-cyclopentyl-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}butanediamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]propanamide
N-cyclopropyl-6-(2-fluoro-5-methoxyphenyl)pyridazin-3-amine
1-({1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
4-cyclopropyl-6-[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyrimidine
(1R,3S)-3-(2-aminoethoxy)-7-[(5-cyclohexylthiophen-2-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
[(3-{2-[4-(2,4-difluorobenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
1-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
N-({7-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
2-cyclopropyl-5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]pyrimidin-4-ol
1-methyl-4-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]morpholine-4-carboxamide
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(2-methoxyacetyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-benzyl-3-methyl-8-[(4-phenylphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
1-(2-methylphenyl)-3-(oxolan-3-yl)-5-(1H-1,2,4-triazol-5-yl)-1H-1,2,4-triazole
N-(1-cyclopentyl-1H-pyrazol-5-yl)-4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carboxamide
4-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-3-(3-methoxyphenyl)-1H-pyrazole
6-(2-aminoethyl)-2-[(3,4-dimethoxyphenyl)methyl]-3,4-dihydropyrimidin-4-one
(2S,4R)-4-(4-{2-[(4-ethylphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
7-chloro-3-(3-hydroxybutyl)-3,4-dihydroquinazolin-4-one
3-methyl-1-[3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
ethyl 4-{3-[(cyclooctylamino)methyl]-6,7-dimethoxyquinolin-2-yl}piperazine-1-carboxylate
5-[5-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
(2R,4R)-N-[2-(3,4-dimethoxyphenyl)ethyl]-4-hydroxy-N-methylpyrrolidine-2-carboxamide
N-(3-phenylprop-2-yn-1-yl)-N-propylpyridine-3-carboxamide
{2-[4-(dimethylamino)-5-methylpyrimidin-2-yl]phenyl}methanol
3-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-3-methyl-1-[4-(pyridin-3-yloxy)phenyl]urea
(3S,4S)-1-[2-(4-acetylphenoxy)acetyl]-4-propylpyrrolidine-3-carboxylic acid
2-({2-amino-6-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
(3R,4S)-4-[ethyl({[4-methoxy-3-(methoxymethyl)phenyl]methyl})amino]oxolan-3-ol
3-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-N,N-dimethylpropane-1-sulfonamide
3-[1-(2-methyl-1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-5-(propan-2-yl)-1,2-oxazole
N-{[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
5-cyclopropyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
N-[2-(morpholin-4-yl)butyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-5-propyl-1,2-oxazole-3-carboxamide
6-[(2-methoxyphenyl)methyl]-2-(4-{[methyl(propan-2-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
7-chloro-4-methyl-2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]quinoline
5-methyl-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,3,4-oxadiazol-2-amine
3-(4-methyl-1,3-thiazol-5-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine