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(2R,3R)-1'-[(2-hydroxypyridin-4-yl)methyl]-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-1H-1,2,3-benzotriazole-5-carboxamide
3-(azetidine-1-carbonyl)-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}benzene-1-sulfonamide
3-benzyl-8-[(3-methoxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-4-[4-(thian-4-yl)piperazine-1-carbonyl]pyridin-2-amine
(1S,5R)-6-(2-methoxyethyl)-3-[1-(4-methoxyphenyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonane
4-(4-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]butan-1-one
1-ethyl-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
1-{3-[2-(3,5-dimethyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
4-methyl-6-(naphthalen-1-yl)pyrimidin-2-amine
2-(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
1-(2-phenylazetidin-1-yl)-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
N-(1-oxo-2,3,4,9-tetrahydro-1H-carbazol-7-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-(4-chlorophenyl)-N-[(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)methyl]cyclopropane-1-carboxamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(2S)-3-methylbutan-2-yl]benzamide
4-(6-ethylpyrimidin-4-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(1-cycloheptylpiperidin-3-yl)-2-(dimethylamino)acetamide
2-[(3-methoxyphenyl)methyl]-8-[2-(1H-1,2,4-triazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
4-cyclohexanecarbonyl-7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1,4-oxazepane
3-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-sulfonyl}-N-methylbenzamide
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-(3-methyl-2-oxoimidazolidin-1-yl)acetamide
4-(1-ethyl-1H-1,2,4-triazol-5-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,3-benzothiazole
3-[2-(2-hydroxyethoxy)ethyl]-1-(1-methyl-4-phenyl-1H-pyrazol-5-yl)urea
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
[1-(4-{4-[(3-phenylpropyl)amino]piperidin-1-yl}benzoyl)piperidin-3-yl]methanol
1-[(3-{[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N-ethyl-2-[4-(furan-2-carbonyl)morpholin-3-yl]-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
(isoquinolin-5-ylmethyl)(methyl)[3-(methylsulfanyl)propyl]amine
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(1-methylpiperidin-2-yl)methyl]amine
4-methoxy-2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}phenol
N-(1-benzothiophen-2-ylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-amine
(1S,3R)-3-amino-N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]cyclopentane-1-carboxamide
6-(benzyloxy)-1-cyclohexyl-4-[3-(pyridin-2-yl)propanoyl]-1,4-diazepan-2-one
N-[(2,4-dichlorophenyl)methyl]-5-ethyl-N-methyl-1,3,4-oxadiazol-2-amine
1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-4-[(dimethylamino)methyl]azepan-4-ol
N-ethyl-2-(4-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperazin-1-yl)acetamide
1-(2-hydroxy-3-{2-methoxy-4-[({[3-(methylsulfanyl)phenyl]methyl}amino)methyl]phenoxy}propyl)piperidin-4-ol
N-[2-(dimethylamino)ethyl]-5-(pyridin-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)(4,4,4-trifluorobutyl)amine
5-(3-fluoro-4-methylphenyl)-1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazole
8-chloro-2-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}quinoline
3-(2,4-dimethoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
5-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol
3-amino-N-(2,4-dichloro-3-methylphenyl)pyrrolidine-1-carboxamide
N-(2-methoxyethyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
methyl 3-[(3-chlorophenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3R,7S,8aS)-7-{[(4-tert-butylphenyl)methyl]amino}-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione