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1-{3-[(4-methylpiperazin-1-yl)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
methyl 3-(2,3-dimethylbenzamido)-6-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
N,2-dimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-[2-amino-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
5-(4-methyl-1,3-oxazol-5-yl)-3-(thiophen-3-ylmethyl)-1,2,4-oxadiazole
1-[1-(3-carbamoylpropanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3,5-dimethyl-4,5-dihydro-1,2-oxazole
5-(2-{4-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3,4-thiadiazol-2-amine
8-chloro-2-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}quinoline
N-{[4-(2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]methyl}-4-methylaniline
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
2-{4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-N-ethylpyridine-4-carboxamide
4-(4-benzyl-5-{[(4-fluorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)-1-(furan-2-ylmethyl)piperidine
2-(cyclopentylmethyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
methyl 1-[(3S,5S)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-[(2-methylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
(cyclohex-3-en-1-ylmethyl)({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
N-[(3R,4S)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
3-methyl-1-[(3-methylphenyl)methyl]-4-(1,8-naphthyridine-2-carbonyl)piperazin-2-one
({5-[1-(1-benzofuran-3-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(3-fluorophenyl)urea
2-ethyl-N-[3-(1H-indol-1-yl)propyl]-4-methyl-1,3-thiazole-5-carboxamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-2-yl)ethan-1-one
2-(2-aminoethyl)-N,5,6-trimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
9-(1-hydroxynaphthalene-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
2-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-5,6-dimethylpyridine-3-carbonitrile
6-tert-butyl-1-methyl-N-[3-(oxolan-3-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(3-hydroxyphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
6-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-2-carbonitrile
1-[2-(methylamino)pyridine-4-carbonyl]-N-(2-phenylethyl)piperidine-4-carboxamide
(3S,4R)-1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]urea
1-(3-chlorophenyl)-4-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]piperazine
6-[4-(1-benzylpiperidin-4-yl)piperazin-1-yl]-9H-purine
[(3-fluoro-2-methoxyphenyl)methyl](methyl){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
4-methoxy-6-[4-(pyrrolidine-1-carbonyl)phenyl]pyrimidine
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(pyridin-2-ylmethyl)piperazine
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
4-[(3-fluorophenyl)methyl]-2-(2-methoxyethyl)morpholine
6-(2,4-dichlorophenyl)-N,N-dimethylpyrimidin-4-amine
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(1H-1,2,4-triazol-3-yl)benzamide
2-(2,4-dichlorophenoxy)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
(1S,6R)-9-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
(1S,5R)-3-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(5-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}furan-2-yl)benzonitrile
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
4-chloro-N,1,5-trimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-3-carboxamide
2-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]benzonitrile
N-cyclopropyl-5-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide