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(3R,9aR)-8-(4-methylbenzenesulfonyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
2-[(5-carboxy-2-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]amino}acetamide
1-ethyl-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylpiperidin-4-amine
3-methyl-4-(1H-pyrazol-3-yl)benzoic acid
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-oxo-3,4-dihydrophthalazine-1-carboxamide
8-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-hydroxy-3-{2-methoxy-4-[({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amino)methyl]phenoxy}propyl)piperidin-4-ol
[3-(1H-imidazol-1-yl)propyl](propyl)(pyridin-4-ylmethyl)amine
2-[(1S,5R)-6-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methyl-1H-1,3-benzodiazole-4-carboxamide
5-(4-fluorobenzoyl)-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5,7-dimethyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]pyrido[2,3-d]pyrimidin-4-amine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
N-[2-(dimethylsulfamoyl)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
4-(3-{[(2,3-dimethylphenyl)methyl]amino}propanamido)benzamide
ethyl 4-{1-[1-(furan-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-1H-pyrazole-3-carboxylate
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-chloro-5-(piperidin-1-yl)benzamide
4-(1-butyl-1H-imidazol-2-yl)-N-(2,5-difluorophenyl)piperidine-1-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
3-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamido]propanamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-4-(1H-1,2,4-triazol-1-yl)butanamide
4-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine-1-carboxamide
(2R)-2-[5-(2-cyclopentylethyl)-4-phenyl-1H-imidazol-1-yl]propanamide
N-(furan-3-ylmethyl)-N-methyl-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
5,6-dimethyl-2-{2-oxo-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydropyridazin-3-one
(4aS,7aR)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-(4-fluorobenzoyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-benzyl-8-(oxane-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclohexyl-3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carboxamide
{3-ethyl-1-[(4-methoxyphenyl)methyl]piperidin-3-yl}methanol
2-{5-[2-(azocan-1-yl)ethyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
(3R,9aR)-8-[(2-fluorophenyl)methyl]-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-(1-ethylpiperidin-4-yl)ethan-1-one
2-methyl-1-{[5-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrrolidine
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-methyl-1-benzofuran-5-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-(6-aminopyridin-3-yl)-2-(4-benzylpiperidin-1-yl)acetic acid
4-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-3-fluorophenol
3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
(3S,4S)-1-(6-methyl-2-phenylpyrimidin-4-yl)-4-(piperidin-1-yl)pyrrolidin-3-ol
(3R,4R)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
4-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
1-(2,5-dihydro-1H-pyrrole-2-carbonyl)-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-(4-chlorophenyl)-4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(3-ethoxypropanoyl)-1-(4-methylphenyl)piperazin-2-one