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3-[(3R,4S)-1-[(2,4-difluorophenyl)carbamoyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
3-(5-methylthiophen-2-yl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1H-pyrazole-5-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
5-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
1-{3-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}ethan-1-one
8-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-({5-[hydroxy(phenyl)methyl]-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-(2-methoxyphenyl)-4-(4-methoxyphenyl)-3-oxopiperazine-1-carboxamide
3-(2-chloropyridine-4-carbonyl)-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-cyclopropyl-1-[1-(4-fluorobenzoyl)piperidin-4-yl]piperidine-3-carboxamide
6-(2-chlorophenyl)-N-ethyl-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-{5-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
3-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-2-(thiophen-2-ylmethyl)propan-1-ol
3-({2-[1-(5-methylthiophene-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-fluoro-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyridine-4-carboxamide
(1R,7S)-3-(4-fluorophenyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
9-[2-(4-fluoro-2-methylphenyl)acetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-hydroxyethyl)-1-{1-[(3-phenoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
4-methyl-N-[2-(4-sulfamoylphenyl)ethyl]-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
2,3,5-trimethyl-N-[3-(morpholin-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)(1H-pyrazol-3-ylmethyl)amine
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,4-dithiepan-6-amine
9-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-6-oxa-9-azaspiro[4.5]decane
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(carboxymethyl)pyrrolidine-3-carboxylic acid
8-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[(dimethylamino)methyl]-1-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-3-ol
N-[(2,3-difluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-{3-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-[(4-methylphenyl)methyl]pyrrolidin-2-one
2-[4-(3-methylphenyl)piperazin-1-yl]-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-(furan-3-ylmethyl)-1-methylurea
2-cyclopropanecarbonyl-8-(6-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-cyclopropanecarbonyl-1'-[(1-methyl-1H-indol-6-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridine
(4aS,8aR)-6-[2-(4-fluorophenoxy)acetyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
4-{[6-(pyrimidin-5-yl)pyridin-3-yl]methyl}morpholine
[(3-{1-[(5-chlorothiophen-2-yl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)methyl]dimethylamine
N-(cyclopropylmethyl)-2-(hydroxymethyl)-N-(2-methoxyethyl)-1H-1,3-benzodiazole-5-carboxamide
methyl (2S,4R)-4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-amido)-1-methylpyrrolidine-2-carboxylate
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(dimethylcarbamoyl)propanoyl]piperidine-3-carboxylate
2-[4-(adamantan-2-yl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
4-[3-(ethoxymethyl)-5-(3-phenylpropyl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
N-(2-ethoxyphenyl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
ethyl({[4-(1H-imidazol-1-yl)phenyl]methyl})(oxan-4-ylmethyl)amine
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyrrolidin-1-yl)propan-1-one
4-{[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-6-yl]formamido}-N-methylbutanamide
N-(4-chloro-3-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}phenyl)acetamide
6-[1-(2-methoxypyridine-4-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol