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[(3R,4R)-4-(azepan-1-ylmethyl)-1-(5-methyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]methanol
4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-3-amine
6-{[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
(2S,4R)-1-(adamantan-2-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
2-(3-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}phenyl)ethan-1-amine
1-(2-chlorophenyl)-3-{1-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-[2-(3-fluorophenyl)piperidin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
5-{2-[1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-oxazol-3-ol
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl](4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
ethyl 4-({[7-fluoro-2-oxo-1-(pyridin-3-ylmethyl)-1,2-dihydroquinolin-3-yl]methyl}amino)piperidine-1-carboxylate
N-(2-methoxyethyl)-1-[1-(pyrimidin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-{1-[1-(1H-indole-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
5-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(butan-2-yl)[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](pyridin-3-ylmethyl)amine
2-{1-[2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzenesulfonyl]azetidin-3-yl}pyridine
4-(hydroxymethyl)-1-(1-methyl-4-phenylpiperidine-4-carbonyl)azepan-4-ol
(1S,5R)-3-benzoyl-6-[2-(difluoromethoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(methylamino)pyridine-4-carboxamide
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}azetidine-2-carboxylic acid
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-methyl-2-(thiophen-2-ylformamido)propanamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]pyridin-2-amine
5-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-N-propylpyrimidin-2-amine
7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1-methyl-1H-imidazol-2-yl)ethyl]benzamide
6-(1H-imidazol-1-yl)-2-methylquinolin-4-ol
1-[2-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-4-ol
8-methoxy-N-[(3-methyloxetan-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}pyridine-3-carboxylic acid
(2S,4S)-4-amino-N-ethyl-1-{2-[4-(3-methylphenyl)piperazin-1-yl]acetyl}pyrrolidine-2-carboxamide
1-(2-methoxyphenyl)-N-[1-(1,3-thiazol-5-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-2-one
5-[2-oxo-2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N3-cyclohexyl-1-cyclopropyl-N5-[(2,4-dimethoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
6-methyl-2-{1-[2-methyl-2-(morpholin-4-ylmethyl)propyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
6-ethoxy-3-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
(2S,3R)-2-amino-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methoxybutan-1-one
3-{5-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)amino)methyl]thiophen-2-yl}prop-2-yn-1-ol
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)pyrrolidin-3-yl]acetamide
1-(prop-2-en-1-yl)-N-[3-(pyridin-4-yl)propyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[7-(3-cyano-2-methoxypyridin-4-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
5-amino-4-chloro-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-1H-pyrazole-3-carboxamide
3-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridin-2-amine
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
(1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}pyrrolidin-3-yl)methanol
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-6-methylimidazo[2,1-b][1,3]thiazole
(3R,9aR)-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(5-methylfuran-2-yl)-N-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide