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3-(4-chlorophenyl)-N-[(methylcarbamoyl)methyl]-3-phenylpropanamide
2-[(1S,5R)-3-[(2-ethoxyphenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-(2-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)-1H-imidazole-2-carboxamide
4-(3-aminothiophene-2-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-(1-{6-[(2-hydroxyethyl)(methyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
(3aR,6aR)-2-(2-methoxyethyl)-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(furan-3-ylmethyl)-4'-(3-methoxypropyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-benzoyl-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(4S)-N-[(4-chlorophenyl)methyl]-4-hydroxy-3,3,4-trimethylpiperidine-1-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(1-methylpiperidin-4-yl)acetamide
(1R,3R,5S)-8-(3,5-difluoropyridine-2-carbonyl)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane
N,2-dimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
2-(2-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)acetic acid
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(3-methoxybenzoyl)piperazine
1-amino-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)cyclopropane-1-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methyl-1H-pyrrole-2-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)quinoline-2-carboxamide
4-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]pyridin-2-amine
(1S,5R)-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-5-methoxy-4H-pyran-4-one
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
8-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{5-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
3-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carboxamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(thiophen-2-yl)azetidine
5-benzoyl-N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{9-[(4-chlorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
3-(1H-imidazol-2-yl)-1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperidine
1-[2-(dimethylamino)-6-(pyridin-2-ylmethyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
5-methoxy-1-methyl-2-[4-(pyrazin-2-yl)piperazine-1-carbonyl]-1H-indole
(2S,4S)-1-benzyl-N-ethyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl){[4-(pyrimidin-5-yl)phenyl]methyl}amine
2-(3-methoxyphenoxy)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-(1-methanesulfonylpiperidin-4-yl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-({2-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(3-fluorophenyl)methyl]-4-(4-methoxyphenyl)-2-methyl-5-oxopiperazine-1-carboxamide
2-fluoro-4-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}phenol
(3S,4S)-1-[(5-methylfuran-2-yl)methyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-[3-(pyridin-4-yl)propanoyl]-1,4-diazepan-2-one
3-({[(3-fluorophenyl)methyl]amino}methyl)-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
{5-fluoro-7-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-7-(propan-2-yloxy)-2H-chromen-2-one
1-methyl-4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazine
4-(1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl)morpholine
1-tert-butyl-N-methyl-5-oxo-N-(quinoxalin-2-ylmethyl)pyrrolidine-3-carboxamide
6-(azepan-1-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine