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7-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-{6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridazin-3-yl}thiomorpholine
2-benzyl-8-(1-methylazepane-2-carbonyl)-2,8-diazaspiro[4.5]decan-1-one
2,4-dimethoxy-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
N-[2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)quinolin-5-yl]acetamide
2-(2,5-dimethylphenoxy)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)propanamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
4-{1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-4-yl}thiomorpholine
3-(4-{1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl}pyridin-2-yl)phenol
8-{4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butanoyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methylpyridine-3-carboxamide
(2S)-1-[(2,3-dimethoxyphenyl)methyl]-4-methyl-2-phenylpiperazine
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
7-methoxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]methanesulfonamide
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-(4-fluorophenyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}azetidine
5-cyclopropanecarbonyl-1'-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{[1-(1,4-oxazepan-4-yl)-1-oxopropan-2-yl]sulfanyl}-3,4-dihydroquinazolin-4-one
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl][(2,4,6-trimethoxyphenyl)methyl]amine
6,6-dimethyl-1-(4-methylphenyl)-N-[(6-methylpyridin-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-4-[4-(propan-2-yl)phenyl]butan-1-one
(1R,2S,9R)-11-(2-ethylbenzoyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-propylpiperazine
1-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-hydroxyethan-1-one
9-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenoxy}-1-(piperidin-1-yl)ethan-1-one
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]butan-1-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(4-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(piperidine-1-carbonyl)piperidine
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-2-(methoxymethyl)piperidine
1-[(3aR,6aR)-3a-(4-propylpiperazine-1-carbonyl)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-methoxyethan-1-one
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-ethyl-N-(2-methylprop-2-en-1-yl)-1,2-oxazole-3-carboxamide
5-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(pyridazine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(3-chlorophenyl)-4-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}piperazin-2-one
3-methyl-3-(4-{1-[(4-methylphenyl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)-1λ6-thiolane-1,1-dione
N-{1-[4-(3-chlorophenyl)-5-[(cyclohexylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}acetamide
8-(3-methylbutanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(1H-imidazol-2-ylmethyl)-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(2-chlorophenyl)methyl]-3-{1-[2-(1H-imidazol-1-yl)acetyl]piperidin-3-yl}propanamide
(4S)-3,3,4-trimethyl-1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-ol
(3S,5R)-N3-(2H-1,3-benzodioxol-5-ylmethyl)-1-benzyl-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
1-methyl-N-{2-[3-(propan-2-yloxy)phenyl]ethyl}-1H-1,3-benzodiazole-5-carboxamide
3-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-N-methylpyridin-2-amine
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
1-({1-cyclohexyl-3-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-5-methyl-1H-1,2,3,4-tetrazole