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8-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(3R,4R)-4-(azepan-1-yl)-1-[(1-ethyl-1H-indol-3-yl)methyl]piperidin-3-ol
N-[2-(pyridin-2-ylsulfanyl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(4aR,8aS)-6-[(2,6-difluorophenyl)methyl]-1-(3,3-diphenylpropyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-[3-(1H-pyrazol-1-yl)azetidin-1-yl]pyridine-3-carboxamide
5-methyl-N-{[1-(phenoxymethyl)cyclopropyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(1S,6R)-9-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethylacetamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3,6-dimethyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-[(2,3-dihydro-1H-inden-2-yl)amino]-N-(2-methoxyphenyl)propanamide
5-({2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}methyl)-N-methylfuran-2-carboxamide
methyl 3-[(3S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
(1H-indol-4-ylmethyl)(methyl)[(5-methyl-1,2-oxazol-3-yl)methyl]amine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(2,4-dimethylphenyl)-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
N-[(1S,2R)-2-aminocyclobutyl]-2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole-4-carboxamide
1-{4-[(4-ethoxypiperidin-1-yl)methyl]-2-methoxyphenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
N,N-diethyl-4-[5-(2-methylpropanoyl)thiophen-2-yl]benzamide
1-{3-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propyl}-1H-pyrazole
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-{[(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
(4aR,7aS)-1-acetyl-4-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-methylbenzene-1-sulfonamide
4-(2H-1,3-benzodioxol-5-yl)-2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]pyrimidine
1-(1-benzoxepine-4-carbonyl)-3-(2-methoxyphenoxy)azetidine
2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(2-methylpropyl)acetamide
4-[(4-fluorophenyl)methyl]-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-pyrazol-1-yl)butan-1-one
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}thian-4-amine
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
1-({4-methyl-5-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
2-(3,4-dimethoxyphenyl)-4-(4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}piperidin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
6-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]pyridine-2-carbonitrile
1-[(3S,4R)-3-cyclopropyl-4-{[5-(trifluoromethyl)pyridin-2-yl]amino}pyrrolidin-1-yl]-2-methoxyethan-1-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(1S,5R)-3-(1-benzofuran-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[2-(dimethylamino)ethyl]-9-(5-propyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
7-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]-4-methyl-1,2-dihydroquinolin-2-one
N-benzyl-3-(2-methyl-1H-imidazol-1-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
9-(2-hydroxybenzoyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
{1-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]piperidin-2-yl}methanol
N-[2-(pyridin-4-yl)ethyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-(cyclopropylmethyl)-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
1,3-dimethyl-2,6-dioxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
[1-(1-methyl-1H-pyrazole-5-carbonyl)-4-(2-phenylethyl)piperidin-4-yl]methanol
(2S)-N2-ethyl-N1-(2-methyl-1-benzofuran-5-yl)pyrrolidine-1,2-dicarboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-N-propyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-[(dimethylamino)methyl]-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]pyrrolidin-3-ol