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2-chloro-4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-methoxyphenol
1-[(3R,4S)-3-(dimethylamino)-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-propoxyethan-1-one
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-3-ol
methyl (2S)-1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
4-{[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]methyl}-N-methylbenzamide
1-[(4-hydroxyazepan-4-yl)methyl]-3-(2-phenoxyphenyl)urea
2-{5-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-phenyl-1H-1,2,4-triazol-3-yl}acetamide
3-({[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
2-(1-{[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(dimethylamino)-4-methyl-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}pyrimidine-5-carboxamide
4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3-(3-methylphenyl)-1H-pyrazole
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
2,4-dimethyl-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)pyrimidine-5-carboxamide
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
5-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
1-cyclopropyl-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}pyrrolidin-2-one
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4-(4H-1,2,4-triazol-4-yl)benzamide
(1S,4S)-2-(2-chlorophenyl)-5-[2-(trifluoromethyl)benzoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N,N-dimethyl-4-({2-[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]-1H-imidazol-1-yl}methyl)oxan-4-amine
(4aR,8aR)-2-methanesulfonyl-7-[3-(2-methoxyphenoxy)propyl]-decahydro-2,7-naphthyridin-4a-ol
1-{2-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}piperidin-2-one
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(6-methylpyrimidin-4-yl)piperidine-4-carboxylic acid
4-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamido]butanoic acid
(2R,6R)-4-(6-aminopyridine-3-carbonyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
1-({5-[(2-aminopyridin-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
1-{2-[(naphthalen-1-yl)carbamoyl]ethyl}-5-oxopyrrolidine-3-carboxylic acid
4-[4-(2,4,6-trimethylphenyl)phenyl]piperidin-4-ol
methyl 3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
1-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzoyl]-4-(1H-imidazol-2-yl)piperidine
1-(3-chlorophenyl)-4-[3-(4-hydroxyphenyl)propanoyl]-5-methylpiperazin-2-one
(3S,4R)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-phenoxypropanamide
2-oxo-8-[4-(pyrrolidin-1-yl)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(3-methyl-1,2,4-thiadiazol-5-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
2-chloro-4-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-6-methoxyphenol
[(3S,5R)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-phenyl-1H-imidazole-4-carboxamide
N-[(3-chlorophenyl)methyl]-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-(3-methoxypyrrolidine-1-carbonyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
2-[4-(adamantan-2-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
3-[(4-hydroxypiperidin-1-yl)methyl]-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-(2-aminoethyl)-N-{[3-(difluoromethoxy)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[4-(4-carbamoylpyridin-2-yl)phenyl]acetic acid
1-[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-2-(1-ethylpiperidin-4-yl)ethan-1-one
4-[(2-hydroxyethyl)sulfamoyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide