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3-(pyrrolidin-1-yl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
(2R)-2-amino-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-phenylacetamide
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
N,N-diethyl-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-cyclopentyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)propanamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(2-chlorophenoxy)piperidine
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(pyridin-3-yl)propanamide
2-{3-chloro-4-[(4-fluorophenyl)methoxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
3-(1-methyl-1H-pyrrol-2-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
4-[(2-ethylpyrimidin-4-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2-hydroxyphenyl)-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-pyrazole-5-carboxamide
1-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
N-ethyl-6-methyl-2-(4-methylphenoxymethyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-methyl-N-{1-oxaspiro[4.5]decan-3-yl}-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N1-[4-(3-methoxyphenyl)phenyl]-N2-methylpyrrolidine-1,2-dicarboxamide
(2R)-2-amino-3-(1H-indol-3-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
9-(1H-imidazol-4-ylmethyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
7-(2-{[(dimethyl-1,2-oxazol-4-yl)methyl]amino}propoxy)-2H-chromen-2-one
1'-[(1-propyl-1H-imidazol-2-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
1-[3-oxo-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decane-8-carbonyl]cyclopropane-1-carboxamide
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]urea
2-[2-(4-chlorophenyl)morpholin-4-yl]quinoline-4-carboxylic acid
N-methyl-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}-N-(3-phenoxypropyl)acetamide
2-(5-{[(dimethylcarbamoyl)amino]methyl}-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl)acetic acid
2-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)-6-methylpyridine
1-(2-fluorobenzoyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
ethyl 4-[6-(1-methylpiperidin-4-yl)pyrimidin-4-yl]piperazine-1-carboxylate
1-methanesulfonyl-4-{4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}piperidine
2-[methyl({[5-(3-phenyl-1,2,4-oxadiazol-5-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl})amino]ethan-1-ol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(5-{1-[3-(1H-pyrazol-5-yl)phenyl]-1H-imidazol-2-yl}furan-2-yl)methanol
8-chloro-2-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)quinolin-4-ol
4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]morpholine-2-carboxamide
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-4-(trifluoromethyl)pyrimidin-2-amine
ethyl 2-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]amino}acetate
2-chloro-5-acetamido-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}benzamide
8-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-[5-({3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)pyrimidin-2-yl]morpholine
1-methyl-9-(2-methyloxolane-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
3-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-4-methylbenzamide
N-{[1-(2-methylpyridine-3-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
4-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-4-oxobutanamide
4-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]benzoic acid
1-cyclopentyl-4-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]piperazin-2-one
2-methyl-2-{4-[2-(propan-2-yl)-1H-imidazol-1-yl]phenyl}propanamide
N-(2-methylprop-2-en-1-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide