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7-chloro-3-({[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)-1,2-dihydroquinolin-2-one
7-(3,6-dimethylpyrazin-2-yl)-4-(5-ethyl-2-methylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3-methyl-1,2-oxazol-5-yl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
4-benzyl-3-(piperidin-4-yl)-1-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-(1H-imidazol-1-yl)-N-(propan-2-yl)benzamide
{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}[3-(1H-pyrazol-1-yl)propyl](pyridin-4-ylmethyl)amine
N-[(3R,4S)-1-(5,6-dimethylpyrazin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-(methylsulfanyl)-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyridine-3-carboxamide
3-(1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazole
4-[(2,3-difluoro-4-methylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
3-[2-amino-4-methyl-6-({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)pyrimidin-5-yl]propanoic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(4-methylphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-cycloheptanecarbonyl-4-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
6-(2,5-dimethylfuran-3-yl)-8-oxo-N-(2-oxopiperidin-3-yl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
6-[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]pyridine-2-carbonitrile
3-{1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1'-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{1-[1-(furan-3-carbonyl)piperidin-4-yl]ethyl}-4-methylpiperazine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}(furan-2-ylmethyl)(oxolan-2-ylmethyl)amine
3-{[(2-phenoxyethyl)amino]methyl}pyrrolidin-3-ol
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-[(4-methylpiperazin-1-yl)methyl]piperidin-2-one
5-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridine-3-carboxamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-2-(methoxymethyl)piperidine
2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-3-(2-methyl-1H-indol-1-yl)propanamide
4-hydroxy-N,N-dimethyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
(1R,2R,4R)-N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1,3-benzothiazole
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2,2,2-trifluoroethyl)benzamide
N-[3-(4-methanesulfonylphenyl)phenyl]acetamide
N-[2-({4-[2-(1,2-benzoxazol-3-yl)acetyl]morpholin-2-yl}formamido)ethyl]acetamide
6-[4-(pyrrolidin-2-yl)phenyl]pyridin-3-amine
2-methyl-4-(2-methylphenyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperazine
ethyl 4-[(5S,9aS,9bS)-1-oxo-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]-1H-pyrazole-3-carboxylate
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-4-carboxamide
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl){[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}amine
3-methyl-8-(3-methyl-1H-pyrazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}-4-oxo-4H-chromene-2-carboxamide
1-(azepan-1-yl)-3-[3-({[2-(2-fluorophenyl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-[(1-hydroxybutan-2-yl)sulfamoyl]-N-[(5-methylpyrazin-2-yl)methyl]benzamide
(1S,6R)-9-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]acetamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(cyclopropylmethyl)propanamide
3-methyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}quinoxalin-2-amine
ethyl 4-(cyclopropylmethyl)-1-(2-cyclopropylquinoline-4-carbonyl)piperidine-4-carboxylate
2-[1-(1H-indole-6-carbonyl)pyrrolidin-3-yl]benzoic acid
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide