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(3aS,6aS)-2-(ethanesulfonyl)-5-(3-phenylpropanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,5R)-3-[(3-chloro-2,4-difluorophenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{5-[3-(4-chlorobenzoyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-(adamantan-1-yl)-N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]acetamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(oxolane-3-carbonyl)piperidin-4-yl]oxy}benzamide
7-(2-hydroxyethyl)-2-{2-[4-(hydroxymethyl)phenyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
6-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]quinoline
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(pyrrolidine-1-sulfonyl)piperidine
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(3-fluorophenoxy)ethan-1-one
1,9-dimethyl-4-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-1,4,9-triazaspiro[5.5]undecane
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-(pyridin-4-ylsulfanyl)acetamide
1-[(5-cyclopentylthiophen-2-yl)methyl]pyrrolidin-3-amine
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-(methoxymethyl)-N-methyl-1,3,4-oxadiazole-2-carboxamide
5-ethyl-N-(1H-indol-6-ylmethyl)-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(cyclohexylmethyl)-4-oxo-N-(propan-2-yl)-5-(thiomorpholine-4-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-[6-(2-methoxyphenyl)pyridazin-3-yl]-2-methylphenol
2-(2-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}ethyl)pyridine
3-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}-1H-pyrazol-1-yl)propanoic acid
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
5-ethyl-1'-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidine
(3R)-N-(3-carbamoyl-2-methylphenyl)-3-hydroxypyrrolidine-1-carboxamide
2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-fluoroethyl)acetamide
1-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}piperidin-3-ol
1-{1-[3-(difluoromethoxy)benzoyl]piperidin-4-yl}-2-phenylethan-1-ol
N-(1-ethyl-1H-pyrazol-4-yl)-4-[2-(phenylcarbamoyl)ethyl]piperidine-1-carboxamide
1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
(1S,4S)-2-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]-2-azabicyclo[2.2.1]heptane
5-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)amino)methyl]-2-methoxyphenol
(1R,5R)-6-benzyl-3-(3-fluorobenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(azepan-1-yl)-2-oxo-N-{[1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]methyl}acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2-chloro-6-fluoro-3-methylbenzoyl)pyrrolidin-3-yl]methanol
1-ethyl-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-(2,4-dimethoxybenzoyl)-7-azaspiro[3.5]nonan-1-ol
2,6-dimethyl-4-({[1-(pyridin-4-yl)propan-2-yl]amino}methyl)phenyl acetate
3-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
4-methoxy-3-(quinolin-3-yl)benzamide
5-{1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
(4aS,8aR)-6-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)cyclohexanecarboxamide
(5-{1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
(2R,3S,6R)-5-(4-methyl-1,3-thiazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-(2-methylpropyl)pyrrolidin-2-one
6-(2-amino-6-methylpyrimidine-4-carbonyl)-3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-(2-methylphenyl)acetamide
3-phenyl-1-(2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)pyrrolidine
2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidine
N-[(4-fluorophenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
2-[4-({8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)phenoxy]acetic acid
2-(dimethylamino)-2-(2-fluorophenyl)-N-(2-hydroxyethyl)-N-propylacetamide