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1-[(5-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-methylpiperazine
3-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-methylpyridin-2-amine
4-benzyl-3-ethyl-1-(6-ethyl-2-methylpyrimidin-4-yl)-1,4-diazepan-5-one
1-ethyl-4-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
(3aR,7aS)-2-[3-(pyrrolidine-1-sulfonyl)thiophene-2-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N,N-dimethyl-4-[4-(1,2-oxazinane-2-carbonyl)phenoxy]piperidine-1-sulfonamide
N-[2-(morpholin-4-yl)ethyl]-4-[4-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)piperidin-1-yl]benzamide
4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3-(propan-2-yl)piperazin-2-one
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(1,4-dioxan-2-ylmethyl)-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
3-{[4-(3-chlorophenyl)-5-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]acetamide
4-(azepane-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)-8-methylquinoline
4-{4-[(2,4-difluorophenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(cyclopropylmethyl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidine-3-carboxylic acid
N-[2-(2-methoxypyridin-3-yl)-4-methylphenyl]propanamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N5-ethyl-N3-methyl-1-(2-methylpropyl)-4-oxo-N3-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
8-{[3-(4-chlorophenoxy)phenyl]methyl}-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}-1-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
N-(1-methylcyclopropyl)-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
1-(2,3-dihydro-1-benzofuran-7-carbonyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
1,3-dimethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-benzyl-3-{[(3-chloropyridin-2-yl)amino]methyl}-N-methylpyridin-2-amine
7-(cyclobutylmethyl)-2-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-methyl-4-[(4-phenyl-1,4-diazepan-1-yl)methyl]benzene-1-sulfonamide
(1R,5R)-N,N-dimethyl-6-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(5-methyl-1,3-oxazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5,7-dimethyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
4-{4-[3-(dimethylamino)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxamide
1-[4-(2-methoxy-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenoxy)piperidin-1-yl]ethan-1-one
N-methyl-3-(2-methyl-1H-imidazol-1-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]butanamide
1-(2,6-difluorobenzoyl)-3-[(dimethylamino)methyl]piperidin-3-ol
1-cyclopentyl-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
2-[4-(3-cyano-6-methylpyridin-2-yl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
N-methyl-N-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-2,3-dihydro-1H-inden-2-amine
N-[(3S,5S)-1-(3-ethoxypropanoyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
(1S,3R)-N1-[2-(2-chlorophenoxy)ethyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
(1S,6R)-9-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3,9-diazabicyclo[4.2.1]nonane
N-cyclopropyl-1-{1-[6-(methoxymethyl)pyrimidin-4-yl]piperidin-4-yl}piperidine-3-carboxamide
(2R)-2,5-diamino-1-(3,3-diphenylpiperidin-1-yl)pentan-1-one
3-{[(5-methylthiophen-2-yl)methyl]carbamoyl}pyridin-1-ium-1-olate
(2R,6S)-4-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-2,6-dimethylmorpholine
6-[(2-butyl-1H-imidazol-4-yl)methyl]-1-propyl-3-[4-(1H-pyrazol-1-yl)phenyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-(4-methoxyphenyl)-3-phenyl-1-[4-(pyrazin-2-yl)piperazin-1-yl]propan-1-one
[1-(1,2-oxazole-3-carbonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol