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2-(3-methoxyphenyl)-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
5-(2-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2S,4S)-1-[(3-phenoxyphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
1-(2-methoxybenzoyl)-4-[6-(methoxymethyl)pyridine-2-carbonyl]piperazine
3-{[(prop-2-en-1-yl)(pyridin-3-ylmethyl)amino]methyl}-4H-chromen-4-one
N-(furan-2-ylmethyl)-1-phenyl-N-(prop-2-en-1-yl)cyclopropane-1-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(2-phenoxyphenyl)ethyl]acetamide
3-(2-methyl-1,3-thiazol-4-yl)-5-(oxolan-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
1-propanoyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
4-(4-{2-methyl-7-oxo-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-6-yl}piperidin-1-yl)-1λ6-thiane-1,1-dione
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-3-(1-methylpiperidin-3-yl)propanamide
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-{1-[1-(4-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
2-(2-methylphenyl)-5-{1-[2-(oxan-2-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
dimethyl[(5-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}furan-2-yl)methyl]amine
1-{3-[2-(furan-2-yl)azepan-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-decahydro-1,6-naphthyridin-2-one
4-(1H-1,3-benzodiazol-1-yl)-1-(3-cyanopyridin-2-yl)piperidine-4-carboxylic acid
(1R,5R)-6-{[4-(2-hydroxyethoxy)phenyl]methyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-acetyl-N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]thiophene-3-carboxamide
N4-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-6-methylpyrimidine-2,4-diamine
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
8-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-amino-4-[1-(2-methoxyethyl)piperidin-4-yl]-5H,6H,7H,8H,9H-cyclohepta[b]pyridine-3-carbonitrile
methyl 3-(5-methylthiophene-2-amido)-6-(piperidin-1-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-N-(2-methylpropyl)propanamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-{1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}azepane
6-(2-methylbutan-2-yl)-N-(4H-1,2,4-triazol-4-yl)-1-benzothiophene-3-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2,6-dimethylquinoline-3-carboxamide
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,3-dihydro-1H-indene-5-carboxamide
N-[(2-ethoxyphenyl)methyl]-6-methyl-4-oxo-N-(prop-2-en-1-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-cyclopropanecarbonyl-N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide
3-[(3S,4R)-4-(morpholin-4-yl)-1-(pyridin-2-ylmethyl)piperidin-3-yl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}propan-1-one
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(4S)-4-hydroxy-3,3,4-trimethyl-N-(thiophen-2-ylmethyl)piperidine-1-carboxamide
2-(2-chloro-4-{[methyl(oxan-4-ylmethyl)amino]methyl}phenoxy)propanoic acid
2-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-butyl-8-(2-methoxypyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]cyclohexanecarboxamide
2-(4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-[(4-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
2-(cyclopropylmethyl)-9-[6-(methoxymethyl)pyridine-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
{4-[2-(methylsulfanyl)pyrimidin-4-yl]phenyl}methanol
6-methyl-5-[5-(quinolin-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(oxolan-2-ylmethyl)benzamide
8-(9H-fluoren-2-ylmethyl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
(2R,6R)-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(2-methoxyethyl)-2-(3-methylbutanoyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide