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(1R,4S)-N-[(2-chloropyridin-3-yl)methyl]-N,1,7,7-tetramethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
3-methyl-1-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2-dihydroquinoxalin-2-one
3-(3-methoxyphenyl)-N-[1-(3-methylpyridin-2-yl)propyl]-1H-pyrazole-4-carboxamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
7-(1-benzothiophen-3-yl)-4-(5-methylthiophene-2-carbonyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methyl-N-{[1-(phenoxymethyl)cyclopropyl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
8-methoxy-N-{[5-(methoxymethyl)furan-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
N3-[(3,4-dimethoxyphenyl)methyl]-N3-methyl-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(methylsulfanyl)acetamide
3-[2-(4-aminopiperidin-1-yl)-2-oxoethyl]-3-benzyl-1-methyl-2,3-dihydro-1H-indol-2-one
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl){[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
4-(benzyloxy)-1-(2-fluoro-6-methoxybenzoyl)piperidine
(2S)-N-[4-(3-fluorophenyl)phenyl]-1-[3-(1H-imidazol-1-yl)propyl]pyrrolidine-2-carboxamide
2-(5-fluoro-2-methylphenyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
2-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
6-oxo-N-[2-(3-phenylpropoxy)phenyl]piperidine-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]acetamide
N-(4-{[1-(1H-1,3-benzodiazol-2-yl)ethyl]carbamoyl}phenyl)-2-methylfuran-3-carboxamide
2-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
1-benzyl-8-[(5-ethylfuran-2-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenylazepane
1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-4-(1,3-thiazol-2-yl)piperazine
4-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
1-(4-{2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-oxoethoxy}phenyl)propan-1-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
(2S,4S)-4-(2,5-dimethylfuran-3-amido)-N-ethyl-1-(2-methoxyethyl)pyrrolidine-2-carboxamide
[(3R,4R)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
3-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-(6-fluoropyridin-3-yl)urea
2-(5-fluoro-2-methoxyphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
(1S,5R)-3-(2H-1,3-benzodioxole-5-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4S)-1-(1H-indol-4-ylmethyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1'-(dimethyl-1,2-oxazole-4-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-butyl-6-methoxy-2-oxo-N-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3S,4R)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-[4-(3,5-dimethyl-1-benzofuran-2-carbonyl)-1,4-diazepan-1-yl]-1,3-benzothiazole
4-(1-methyl-5-{[(4-methyl-1,3-thiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-3-yl)pyridine
(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}-3-propylpiperidin-3-yl)methanol
8-(morpholine-4-sulfonyl)-2-(1,3-thiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
2-[(3-methoxyphenyl)methyl]-8-(1-methyl-1H-imidazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(1R,6S)-N-(2,6-dichloropyridin-4-yl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
N-[2-(oxan-2-yl)ethyl]-3-(piperazine-1-carbonyl)benzene-1-sulfonamide
1-[(3,4-difluorophenyl)methyl]-N-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-amine
1-[(2-methoxyphenyl)methyl]-N-(3-methylbutyl)-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2,6-dimethyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)pyrimidine-4-carboxamide
(4aR,8aS)-1-[2-(4-methoxyphenyl)ethyl]-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridin-2-one
[1-(2-fluorophenyl)propan-2-yl]({[4-(pyrrolidine-1-carbonyl)phenyl]methyl})amine
2-methyl-6-[1-(pyridin-3-yl)propan-2-yl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-(3-{5-[2-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-1-yl}propyl)pyridin-3-amine
5-cyclobutyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1,3,4-oxadiazol-2-amine