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3-{[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]methyl}-4-propyl-4H-1,2,4-triazole
3-[1-(3-methoxyphenoxy)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
dimethyl({1-[4-({methyl[2-(methylsulfanyl)ethyl]amino}methyl)phenyl]ethyl})amine
3-(3,4-dimethoxyphenyl)-N-(5-oxo-1-phenylpyrrolidin-3-yl)propanamide
4-(3-hydroxyphenyl)-N-[3-(methylsulfamoyl)phenyl]piperidine-1-carboxamide
3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2-methoxyquinoline
{2-oxo-2-[3-(2-phenylacetyl)piperidin-1-yl]ethyl}urea
1-(4-chlorophenyl)-4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
1-(5-chloropyridin-2-yl)-4-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]piperazine
3-[4-(4-methoxyphenyl)butyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
N-(2-methoxyethyl)-2,7-dioxo-N-(pyridin-3-ylmethyl)-1,3-diazepane-4-carboxamide
1-[2-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)phenyl]ethan-1-one
(2S)-2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-phenylpropanamide
(2R)-2-amino-1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-3-methoxypropan-1-one
4-[1-benzyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
(3E)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}hex-3-enamide
N-[3-(1H-pyrazol-3-yl)phenyl]-2H-1,3-benzodioxole-5-carboxamide
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-4-propylpyrimidine-5-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(1H-pyrrol-1-yl)ethyl]amino}methyl)piperidin-2-one
1-{3-[(4-methoxypiperidin-1-yl)methyl]-6-methylquinolin-2-yl}piperidin-3-ol
6-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}pyridine-3-carbonitrile
N,N,4-trimethyl-3-{[(2-methylpropyl)(prop-2-en-1-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(4-chloro-1H-pyrazol-1-yl)-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane-1-carbaldehyde
1-{1'-[(2-ethoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-(furan-3-ylmethyl)-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
9-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-hydroxyethyl)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
N-cyclopropyl-4-(pyridin-4-yl)benzamide
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
1-(1-methyl-1H-pyrazole-4-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3H,4H-pyrido[4,3-d]pyrimidin-4-one
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(thian-4-yl)piperazine
N-(5-propyl-1,3,4-oxadiazol-2-yl)-1-(thian-4-yl)piperidin-4-amine
1-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
4-(5-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}pyrimidin-2-yl)morpholine
[(3-ethoxy-4-methoxyphenyl)methyl](methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-N-[(3S)-piperidin-3-yl]-2,3-dihydro-1H-isoindole-4-carboxamide
N-methyl-4-[5-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-cyclohexyl-N,4-dimethyl-5-{1-[(pyridin-2-ylmethyl)amino]ethyl}pyrimidin-2-amine
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
2-ethyl-9-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
(3S)-1-[(5-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]-3-fluoropyrrolidine
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-indole-5-carboxamide