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2-[(4-chlorophenyl)methyl]-8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
methyl 2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-6-methylpyrimidine-4-carboxylate
(2S,4S)-4-{[(3-chlorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
1-{3-oxo-3-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}piperidine-4-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[3-(3-methoxyphenyl)benzoyl]pyrrolidine-2-carboxamide
(1S,6R)-9-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3,9-diazabicyclo[4.2.1]nonane
2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxylic acid
(4aS,7aR)-1-(3,5-dimethylbenzoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(furan-2-amido)-7-oxo-N-[(4-phenyloxan-4-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-{2-[(4-fluoro-3-methoxyphenyl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-6-methylpyridine
N-ethyl-4-({[(1S,2S)-2-hydroxycyclohexyl]carbamoyl}amino)-N-phenylbenzamide
methyl 1-benzyl-3-(furan-3-amido)-5-[(2-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(1H-imidazol-1-ylmethyl)piperidine
N-cyclopropyl-2-{4-[2-(naphthalen-1-yl)-1H-imidazol-1-yl]piperidin-1-yl}acetamide
(1S,6R)-9-{[2-methoxy-5-oxo-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
5-{2-[5-(6-methyl-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
2-(4-{[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]methyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
3-methyl-4-(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
1-[4-(1H-indol-2-yl)phenyl]-N-(oxan-3-yl)piperidin-4-amine
N-ethyl-N-(2-methylprop-2-en-1-yl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-1-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]urea
4-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidine-1-carbonyl]benzene-1-sulfonamide
1-methyl-1'-[(4-methyl-1H-imidazol-5-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-(2-phenylphenyl)-4-[3-(pyrrolidin-1-yl)propanoyl]piperazin-2-one
9-[2-(3,4-dimethylphenoxy)ethyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{9-[(1-ethyl-1H-imidazol-5-yl)methyl]-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl}-2-(propan-2-yloxy)ethan-1-one
2-cyclopropyl-8-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(cyclopropylmethyl)-3-(1H-imidazol-2-yl)-N-(oxolan-2-ylmethyl)benzamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(1-methyl-3-phenyl-1H-pyrazol-5-yl)urea
(1R,2R,6S,7S)-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4-azatricyclo[5.2.1.02,6]decane
4,6,7-trimethyl-2-(4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,4-diazepan-1-yl)quinazoline
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyrazine-2-carboxamide
4-{1-[2-(3-methylpyridin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-2,1,3-benzoxadiazole
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
1-{3-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(isoquinolin-1-yl)benzamide
3-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]quinoline-4-carboxylic acid
3-({2-[1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}propanoic acid
(3R)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
4-(naphthalen-2-yloxy)-1-(pyridin-4-yl)piperidine-4-carboxylic acid
N,N-diethyl-15-methyl-13-oxo-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
benzyl 3-(1-cyclopropyl-1H-pyrrole-2-amido)pyrrolidine-1-carboxylate
[3-(methylsulfanyl)propyl](pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
2-(1H-indazol-1-yl)-1-[6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl]ethan-1-one
(3S,9aR)-3-[(4-methoxyphenyl)methyl]-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2,4-dichloro-3-methylphenyl)-3-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]urea
2-(dimethylamino)-7-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one