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2-ethyl-4-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-(propan-2-yl)piperazine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]acetamide
2-(4-{[methyl(propan-2-yl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
2-methyl-3-({4-[2-(thiophen-2-yl)azetidine-1-carbonyl]piperidin-4-yl}oxy)pyridine
3-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[3-(benzyloxy)phenyl]-1-(1,4-dioxan-2-ylmethyl)-1-methylurea
[4-(4-methoxyquinazolin-6-yl)phenyl]methanol
N-[(6-methoxypyridin-3-yl)methyl]-N-methylthian-4-amine
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]benzonitrile
2-chloro-N-(2-{[3-(piperidin-3-yl)phenyl]formamido}ethyl)benzamide
(4-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}-1,4-oxazepan-6-yl)methanol
2,6-dimethoxy-4-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenol
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1-(4-methylpiperazin-1-yl)ethan-1-one
1'-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2,6-dimethylpyrimidine-4-carboxamide
2-[3-(5-methylfuran-2-yl)-5-[4-(piperidin-1-ylmethyl)phenyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-cyclopropyl-1-(1-{furo[3,2-c]pyridin-4-yl}piperidin-4-yl)piperidine-3-carboxamide
8-(2,3-dihydro-1H-inden-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(3-fluorophenoxymethyl)-N-(2-methoxyethyl)-N-methyl-1,3-oxazole-4-carboxamide
5-(morpholin-4-yl)-2-(pyrimidin-2-ylmethyl)-2,3-dihydropyridazin-3-one
N-[(3-chlorophenyl)methyl]-3-[1-(oxolan-3-ylmethyl)piperidin-4-yl]propanamide
2-methyl-5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
5-(azepan-1-yl)-1-ethyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
(3R,4S)-4-{4-[(2-methoxynaphthalen-1-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
5-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
benzyl(cyclopropylmethyl){[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}amine
2-{[4-phenyl-5-(2,4,5-trimethoxyphenyl)-1H-imidazol-1-yl]methyl}morpholine
1-(3-methoxyphenyl)-4-[2-(propan-2-ylsulfanyl)ethyl]piperazin-2-one
5-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-(3,5-dimethyl-1-benzofuran-2-yl)-1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1H-1,2,3-triazole
(1S,3R)-N1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
(4aR,7aS)-1-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 4-{2,7-diazaspiro[4.5]decan-7-ylmethyl}-1H-pyrazole-3-carboxylate
2-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-thiazole-4-carboxamide
3-{1-[1-(1-ethylpiperidine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
3-chloro-5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-(6-hydroxy-4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,4-diazepan-1-yl)propane-1,3-diol
5-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carbonyl]-2-methyl-1-phenyl-1H-1,3-benzodiazole
N-[(3,5-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-3-methylpyridine-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(3,4-dihydro-2H-1-benzopyran-3-yl)piperazine
N-{1-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
2-{[3-(3-{furo[3,2-c]pyridin-4-yl}phenyl)-1H-pyrazol-1-yl]methyl}-5-methyl-1,3,4-oxadiazole
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-3-yl)propan-1-one
2-{4-[(3-methoxyphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
3-{[(2-hydroxypropyl)amino]methyl}-6-methyl-1-(prop-2-en-1-yl)-1,2-dihydroquinolin-2-one
4-(1H-pyrazol-4-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)butanamide
(1R,5R)-6-(cyclobutylmethyl)-3-(6-methoxypyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonane
(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
2-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)acetamide
4-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-4H-1,2,4-triazole