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3-(3,4-dimethoxybenzoyl)-1-(1H-1,2,4-triazole-5-carbonyl)piperidine
4-(2,5-dimethoxybenzoyl)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-(furan-2-ylmethyl)-N-methyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
methyl 3-[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]propanoate
(2S,4R)-4-{[(2,6-difluorophenyl)methyl]amino}-1-(2,2-diphenylethyl)-N-methylpyrrolidine-2-carboxamide
N-cyclohexyl-4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)piperidine-1-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(5-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-ylmethyl]-2,1,3-benzoxadiazole
2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pyridine-4-carboxamide
4-(1H-pyrazol-3-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
3-cyclopentyl-N-[(1-ethylpiperidin-3-yl)methyl]propanamide
N-ethyl-5-[3-(propoxymethyl)pyrrolidine-1-carbonyl]pyrimidin-2-amine
{4-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(methyl)amino)methyl]oxan-4-yl}methanol
(3S,4R)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-benzyl-9-[(2S)-2,4-diaminobutanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-fluorophenyl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,4-diazepane
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-imidazol-1-yl)propyl]acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(propane-2-sulfonyl)pyrrolidine-3-carboxylic acid
2-{9-[3-(dimethylamino)benzoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
6-{[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[4-chloro-2-(trifluoromethyl)phenyl]-3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2,3-dihydro-1H-inden-2-amine
(3aS,6aS)-2-cyclopentanecarbonyl-5-(thiophen-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(4-{4-[(furan-2-ylmethyl)amino]piperidin-1-yl}phenyl)-2-phenoxyacetamide
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]-N-[2-(1H-pyrazol-1-yl)phenyl]piperidine-1-carboxamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(1H-pyrazol-3-ylmethyl)amine
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[1-(ethylsulfanyl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
3-{1-[4-(dimethylamino)benzoyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
1-methyl-2-[5-(1H-1,2,4-triazol-5-ylsulfanyl)furan-2-yl]-1H-1,3-benzodiazole
N-(1H-indol-4-ylmethyl)-3-propanamidobenzamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}propan-1-one
(2S,4S)-N-ethyl-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(1H-pyrazole-3-carbonyl)piperidine-3-carboxylic acid
(1S,5R)-3-(2-methyl-1H-pyrrole-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamide
2-[5-(1,1-dioxo-1λ6-thian-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-4-(pyrrolidin-1-yl)butanamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxyphenoxymethyl)piperidine
N-[2-(3-methoxyphenyl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-[(2,3-difluorophenyl)methyl]-4-[1-(furan-2-carbonyl)pyrrolidin-3-yl]piperidine
4-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]piperidin-1-yl}-2-methyl-6-propylpyrimidine
8-[3-(1H-pyrrol-1-yl)propyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1H-1,3-benzodiazole
1-(6-hydroxy-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,4-diazepan-1-yl)-3-methylbut-2-en-1-one
5-methyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1H-pyrazole-3-carboxamide
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
{5-[2-(benzyloxy)ethyl]-1H-indol-2-yl}methanol
[(3,4-dimethoxyphenyl)methyl]({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine