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8-({3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl](methyl)[(1-methylcyclopropyl)methyl]amine
6-fluoro-2-{[4-(oxolan-2-ylmethyl)piperazin-1-yl]methyl}quinolin-4-ol
1-{2-[(5-chloropyrimidin-2-yl)oxy]hex-5-en-1-yl}piperidine-4-carboxylic acid
2-(4-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
1-{1-[1-(4-fluorophenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
methyl 2-[cyclopentyl({[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl})sulfamoyl]benzoate
2-cyclopropyl-9-[3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
(2R,4S)-1-(3,3-diphenylpropanoyl)-4-hydroxypiperidine-2-carboxylic acid
1-(7-chloro-2-methylquinoline-4-carbonyl)piperidin-3-amine
6-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-N-ethyl-N-methylpyridine-3-carboxamide
5-[4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(2-phenoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}thiophene-2-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-benzyl-3-ethyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
N-[3-(2-fluorophenyl)propyl]oxolane-3-carboxamide
3-({1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidin-3-yl}formamido)propanamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(pyrimidin-4-ylmethyl)acetamide
{2-[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]-1,3-thiazol-4-yl}methanol
3-{1-[(3-methyl-1-benzofuran-2-yl)methyl]-1H-1,2,3-triazol-4-yl}piperidine
N-ethyl-2-methoxy-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
2-(6-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}acetamide
(2R,3S,6R)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-2-(methylamino)pyrimidine-5-carboxamide
5-[bis(prop-2-en-1-yl)amino]-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(1-{2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-yl)methanamine
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(4-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}morpholin-3-yl)-N,N-dimethylacetamide
2-[1-(2-fluoroethyl)-4-phenyl-1H-imidazol-5-yl]quinoline
8-(4,6-dimethoxypyrimidin-2-yl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-amino-4-({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}amino)quinazoline-6-carboxylic acid
4-(2,6-dimethylpyridin-4-yl)-N-[2-(propan-2-ylsulfanyl)phenyl]piperazine-1-carboxamide
5-({[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]carbamoyl}amino)-2-fluoro-N-methylbenzamide
3-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
5,7-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
(3R,4R)-4-(hydroxymethyl)-1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperidin-3-ol
2-chloro-4-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[(prop-2-en-1-yl)amino]-N-propylbenzamide
4-(cyclopropylmethyl)-1-(isoquinolin-1-yl)piperidine-4-carboxylic acid
N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(quinoxalin-6-ylmethyl)acetamide
N-{[1-(2,6-dimethylpyridin-4-yl)piperidin-4-yl]methyl}acetamide
4-(1H-1,3-benzodiazol-2-ylmethyl)-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[3-(pyridin-3-yl)propyl]amine
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)furan-2-carboxamide
2-(dimethylamino)-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide