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1-benzyl-4-(isoquinolin-1-yl)-1,4-diazepan-6-ol
N-benzyl-5-(3,4-difluorophenoxymethyl)-N-(2-hydroxyethyl)-1,2-oxazole-3-carboxamide
6-(1-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
N,5-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]pyrazine-2-carboxamide
(5S,9aS,9bS)-5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3aS,6aS)-2-cyclohexyl-5-(1,3-thiazol-5-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-(2,3-dihydro-1H-inden-2-yl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(2-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[2-methoxy-4-({[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
5-[bis(prop-2-en-1-yl)amino]-1-(cyclohexylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
7-(2-methoxyacetamido)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,2,4-trimethylpyrimidine-5-carboxamide
1-(cyclopropylmethyl)-4-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperazine
3-chloro-5-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidine-5-carboxamide
2-methyl-4-propyl-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-[(1-propylcyclobutyl)methyl]-1-(pyridine-3-carbonyl)piperidin-4-amine
N-[(1R,3R)-3-aminocyclopentyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
5-fluoro-2-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}-3-methyl-1H-indole
4-(2-methylphenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-4-carboxylic acid
4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine-1-sulfonamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
4-[7-(pyridine-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
methyl[(4-methyl-1H-imidazol-2-yl)methyl][(1-methylpiperidin-3-yl)methyl]amine
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3-(4-methylphenoxymethyl)piperidine
9-(2-ethoxybenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl[2-(2-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)ethyl]amine
5-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
(2S)-3-(1H-indol-3-yl)-2-({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)propan-1-ol
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-propylacetamide
5-(1H-1,3-benzodiazol-2-yl)-2-methoxyphenol
1-[3-(furan-2-yl)propanoyl]-4-(3-methylphenoxy)piperidine-4-carboxylic acid
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
(3R,4R)-4-amino-1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]piperidin-3-ol
N-[(3S,4R)-1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}propan-1-one
1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
4-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperazine-1-carbaldehyde
N-methyl-4-(4-methylphenoxy)-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
N-[2-(3-ethylphenoxy)ethyl]-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(4-hydroxypiperidin-1-yl)propan-1-one
4-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}piperazin-2-one
3-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
(4aS,8aR)-1-(2-aminoethyl)-6-(5-propylthiophene-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-({1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-2,3-dimethylbenzamide
N,5-dimethyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-1-propyl-1H-pyrazole-4-carboxamide