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2-methyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-4,5,6,7-tetrahydro-1H-indol-4-one
1-{3-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
4-(2,6-dimethylpyridin-3-yl)-N-[1-(furan-2-carbonyl)piperidin-3-yl]pyrimidin-2-amine
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-amido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
4-cycloheptanecarbonyl-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2,2,2-trifluoro-1-{4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxylate
7-[2-(pyridin-4-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-[5-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-(3-chlorophenyl)-4-{[3-(2-hydroxyethoxy)phenyl]methyl}-5-methylpiperazin-2-one
(2R,3R)-3-(dimethylamino)-1'-[(3-fluoro-2-hydroxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(benzyloxy)-8-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
2-methyl-3-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}quinoxaline
2-[2-(1-methylpyrrolidin-3-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxamide
1-(piperidin-3-ylmethyl)-N-[2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-cyclohexyl-N,7,8-trimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-ol
2-amino-3-ethyl-N-(1-methanesulfonylpiperidin-4-yl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[({4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)sulfanyl]pyridine
(1S,5R)-3-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(piperidin-3-ylmethyl)benzoyl]-4-(pyridin-3-yl)piperazine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-[(4-chlorophenyl)methyl]-8-(piperidin-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
(3aR,6aR)-2-acetyl-5-[(8-fluoro-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S)-2-hydroxy-1-(4-{[5-(methylsulfanyl)-4-phenyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)propan-1-one
4-{3-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrole-2-carbonyl]phenyl}-2-methylbutan-2-ol
N,N-dimethyl-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,3-oxazole-4-carboxamide
N-{2-[(6-ethyl-2-methylquinolin-4-yl)formamido]ethyl}pyridine-3-carboxamide
N-({1-[(5-ethylpyridin-2-yl)methyl]piperidin-3-yl}methyl)pyrimidine-4-carboxamide
{[6-(4-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
5-(4-acetylpiperazine-1-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]piperidin-2-one
{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}[(4-methyl-1H-imidazol-5-yl)methyl]amine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[5-(methoxymethyl)furan-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[2-(dimethylamino)ethyl]({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)carbamoyl}pyridin-1-ium-1-olate
2-[1-methyl-4-(5-methyl-1,3,4-thiadiazol-2-yl)-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
N-(3-methylbutyl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3aR,6aS)-5-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3,4-dimethoxyphenyl)ethyl]acetamide
8-methanesulfonyl-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
2-(2-methyl-1,3-thiazol-4-yl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}acetamide
N-methyl-4-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)benzene-1-sulfonamide
[(3R,4S)-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-(1H-indol-3-yl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
6-methoxy-3-[1-(pyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one