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2-[4-(1-benzoxepine-4-carbonyl)morpholin-3-yl]acetamide
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(3-methylpyridin-2-yl)piperazine
2-(butylsulfanyl)-5-(1H-imidazol-2-yl)pyrimidine
N-[2-(1H-imidazol-4-yl)ethyl]-2-(methylamino)pyridine-4-carboxamide
5-chloro-6-[8-(2-hydroxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carboxylic acid
4-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-1,3-diazepane-2,4-dione
3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrrolidine-1-carboxamide
(2R,4R)-4-hydroxy-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)pyrrolidine-2-carboxamide
1-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-3-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)urea
2-(4-{[(4-fluorophenyl)carbamoyl]formamido}-3,5-dimethyl-1H-pyrazol-1-yl)acetic acid
4-(3-hydroxy-3-methylbutyl)-N-(2-oxopyrrolidin-3-yl)benzamide
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(thiolan-3-yl)piperidin-4-yl]oxy}benzamide
(3aR,6aR)-2-(1-benzothiophen-3-ylmethyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-cyclohexyl-2-[3-(pyridin-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-{[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
N-[4-(dimethylcarbamoyl)-2-methylphenyl]-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
7-{[2-(benzylamino)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]furan-2-carboxamide
N-butyl-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
1-benzoyl-2-{1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}piperidine
N'-[2-(methylsulfanyl)phenyl]-N-(oxolan-2-ylmethyl)-N-propylbutanediamide
(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
(2S,4R)-4-amino-N,N-diethyl-1-(4-methyl-1H-imidazole-2-carbonyl)pyrrolidine-2-carboxamide
N-({1-[(4-ethylphenyl)methyl]piperidin-3-yl}methyl)-4-methoxybenzene-1-sulfonamide
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
6-methyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2-fluorobenzene-1-sulfonamide
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]oxolane-2-carboxamide
1-[(3-fluorophenyl)methyl]-4-{[4-(pyridin-2-yl)phenyl]methyl}piperazine
5-(1H-1,3-benzodiazol-2-ylmethyl)-N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl (2S)-1-({4-[1-(2-phenylethyl)piperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)pyrrolidine-2-carboxylate
[(4-ethyl-1,3-thiazol-2-yl)methyl][1-(1H-imidazol-1-yl)propan-2-yl]amine
9-(but-3-yn-1-yloxy)-4-(3-fluorobenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-methoxy-N-[(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-3-yl)methyl]benzene-1-sulfonamide
N-[(3S,4R)-1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-(1,3-benzothiazol-2-yl)-N-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-amine
2-(2,3-difluorophenoxymethyl)-N-methyl-N-[2-(piperidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-4-[(4-phenylphenyl)methyl]piperazin-2-one
1-(3-hydroxy-1,2-oxazole-5-carbonyl)-4-(pyridin-4-yl)-1,4-diazepan-6-ol
1,5-dimethyl-4-{3-methyl-6-oxo-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-4-yl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-(2-methylphenyl)-3-{4-[3-(morpholin-4-yl)propyl]-1,4-diazepan-1-yl}-3-oxopropanamide
benzyl 4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane-1-carboxylate
2-(2H-1,3-benzodioxol-5-yl)-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}acetamide
3-(1-{4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-1H-imidazol-2-yl)pyridine
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-1-phenylpyrrolidin-2-one
1-[(4-fluoro-3-methoxyphenyl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
(1R,9aR)-1-({[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol