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6-fluoro-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[(1-ethyl-1H-indol-3-yl)sulfanyl]-N-[(1-methylpyrrolidin-3-yl)methyl]acetamide
3-(1H-1,3-benzodiazol-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-{[(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)amino]methyl}pyrrolidin-3-ol
ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
3-methyl-7-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-[5-chloro-2-(propan-2-yloxy)phenyl]-1-methyl-1H-1,2,3,4-tetrazole
N-(1,4-dioxan-2-ylmethyl)-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
(3aS,6aS)-2-cyclopentyl-5-(2,3,6-trifluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-(morpholin-4-yl)ethan-1-one
[1-(3-{[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}propyl)piperidin-3-yl]methanol
N-(1H-indol-3-yl)-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
1-(4-methylquinazolin-2-yl)-N-[(1-phenylcyclopentyl)methyl]piperidine-4-carboxamide
(2S,4S)-4-{4-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxylic acid
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(prop-2-en-1-yl)acetamide
3-{[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]oxy}pyridine
1-{imidazo[1,2-a]pyridine-6-carbonyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[(5-methyl-1H-imidazol-4-yl)methyl]benzamide
1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
4-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydrophthalazin-1-one
2-(2-chlorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
9-(cyclopropylmethyl)-1-methyl-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
5-[5-(1-cyclohexanecarbonylpyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]-1-methyl-1,2,3,6-tetrahydropyridine
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}acetamide
2-[({5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}amino)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-(2-fluorophenyl)-2-{3-[3-(pyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
1-{2-[2-(2-chloro-4-fluorophenyl)acetamido]ethyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
8-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
3-cyclopentyl-3-[(2,4-dimethoxyphenyl)methyl]-1-(pyridin-3-yl)urea
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(ethyl)methylamine
1-(ethanesulfonyl)-3-[2-(3-methoxyphenyl)ethyl]piperidine
(4aS,7aR)-1-(2-aminopyridine-4-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aS,6aS)-2-(dimethylcarbamoyl)-5-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-(3-phenoxyphenyl)-1H-1,2,3-triazole
1-(adamantan-1-yl)-4-(1-methyl-1H-imidazole-5-carbonyl)piperazine
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-(methylamino)pyridine-3-carboxamide
N-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-[(4-fluorophenyl)methyl]piperidin-3-amine
methyl 3-[3-(furan-2-yl)propanoyl]-9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-cyclopropanecarbonyl-2-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(2-hydroxyethyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(propan-2-yl)acetamide
4-{3-cyclopropyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1H-1,2,4-triazol-1-yl}-3-methylpyridine
3-(4-benzylpiperazine-1-carbonyl)-6-methyl-1-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-1,4-dihydropyridin-4-one
5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole
2-{4-[3-(pyridin-3-yl)azetidine-1-carbonyl]piperidin-1-yl}acetamide
(1R,5S)-8-(3-phenyl-1H-pyrazole-4-carbonyl)-3,8-diazabicyclo[3.2.1]octane
1-cyclobutanecarbonyl-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)pyridin-2-amine