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2-methyl-N-{1-[1-(4-oxopentanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3,4-dimethoxybenzamide
2-(2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-6-methyl-2,3-dihydropyridazin-3-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)pyrrolidine-3-carboxylic acid
N-[2-(1H-imidazol-4-yl)ethyl]-6-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-hydroxy-N-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}methyl)acetamide
1-{1-[(2-fluoro-4-methylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-2,3-dihydro-1H-isoindole
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidin-2-amine
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
[(2S,4R)-4-(dimethylamino)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl]methanol
7-[(4-hydroxy-4-phenylpiperidin-1-yl)methyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-(4-methanesulfonylphenyl)-1-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazole
2-amino-6-(2-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]-1-(oxolane-2-carbonyl)piperidine
4-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-1λ6-thiane-1,1-dione
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-yl]methanol
(2S)-2-[(6-methoxy-3-methyl-1-benzofuran-2-yl)formamido]-3-(pyridin-4-yl)propanoic acid
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N-ethyl-N-(2-hydroxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-1-methyl-1H-indole-2-carboxamide
N-[(3-methoxyphenyl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,3-benzotriazole-5-carboxamide
1-[1-(2,5-dimethoxybenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
4-ethyl-1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]-1,4-diazepan-5-one
N-(3-fluorophenyl)-3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazole-5-carboxamide
7,7-dimethyl-2-phenyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-6-methylpyrimidin-2-amine
1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[3-(2-fluorophenyl)propyl]-1-(oxan-4-yl)piperidine-3-carboxamide
N-{5-[2-(2,4-dioxoimidazolidin-1-yl)acetamido]-2-methoxyphenyl}benzamide
8-methoxy-N-(4H-1,2,4-triazol-4-yl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-3,5-difluoropyridine-2-carboxamide
(2R,6S)-1-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)-2,6-dimethylpiperidine
[(2E)-3-(furan-2-yl)prop-2-en-1-yl](furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amine
N-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-ol
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-3-azaspiro[5.5]undecan-9-amine
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-{4-[1-(2,5-dichlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
1-cyclopropanecarbonyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-4-carboxamide
7-(3-chlorophenyl)-4-(2,2-dimethyloxane-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}phenyl)formamido]acetamide
N-[3-(4-methylbenzenesulfonamido)propyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
1-[4-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)phenyl]ethan-1-one
1-cyclohexyl-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N,2,3,5-tetramethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclopropyl-1,3-dimethyl-N-{[3-(oxolan-2-ylmethoxy)phenyl]methyl}-1H-pyrazole-5-carboxamide
(1S,5R)-3-(5-phenyl-1,2-oxazole-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one