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N,3,5-trimethyl-N-{[3-(trifluoromethyl)phenyl]methyl}-1H-indole-2-carboxamide
1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}pyrrolidin-2-one
N-(butan-2-yl)-N-methyl-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
6-[(diethylamino)methyl]-N-[(dimethyl-1,3-thiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
diethyl[(3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)methyl]amine
3-methyl-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}urea
1-(3-methoxyphenyl)-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazin-2-one
(4aR,8aS)-1-[2-(4-chloro-2-methylphenoxy)acetyl]-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]pyrrolidine-1-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
1-({5-[(3-cyanophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
(1R,3S)-7-(1-tert-butyl-1H-pyrrole-3-carbonyl)-7-azaspiro[3.5]nonane-1,3-diol
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(1,3-thiazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)pyrrolidine-3-carboxylic acid
3-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}pyridin-2-amine
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[(2-ethoxyphenyl)methyl]-N-ethyl-3-methylfuran-2-carboxamide
1-(2-methoxyethyl)-3-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]piperidine
2-benzyl-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
4-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-1,2-dimethylpiperazine
4-(4-{[2-(dimethylamino)-2-(4-methylphenyl)ethyl]amino}piperidin-1-yl)-6-methylpyrimidin-2-amine
1-(3,5-difluoropyridine-2-carbonyl)-2-methyl-4-(2-methylphenyl)piperazine
(3S,4R)-3-benzyl-4-methyl-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-ol
2-[2-(3-methoxyphenyl)ethyl]-4-[3-(3-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-benzyl-1-methyl-5-[3-(5-methylfuran-2-yl)butyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(4-chlorophenyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)butanamide
3-(2-fluorophenyl)-N-[3-(3-oxopiperazin-1-yl)propyl]-1H-pyrazole-5-carboxamide
N-(1H-1,3-benzodiazol-2-yl)-2-[(2H-1,3-benzodioxol-5-ylmethyl)(cyclopropyl)amino]acetamide
5-[(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)methyl]-1,3-dimethylimidazolidine-2,4-dione
N-[(1-methylpyrrolidin-3-yl)methyl]-3-phenoxybenzamide
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
propan-2-yl 2-chloro-5-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-amido]benzoate
1-{3-[({3-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]propyl}pyrrolidin-2-one
4-{4-[(3,4-difluorophenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-4H-1,2,4-triazole
4-{[3-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
5-cyclopropyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[6-hydroxy-4-(quinolin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
3-methyl-1-[(3-methylphenyl)methyl]-5-(oxan-4-yl)-1H-1,2,4-triazole
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
3-[3-(oxan-4-yl)-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]pyridine
5-[(4,5-dimethylfuran-2-yl)methyl]-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
3-methoxy-N-[(1-methylpiperidin-2-yl)methyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
4-(benzyloxy)-1-(1,3-thiazole-4-carbonyl)piperidine
4-{1-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carbonyl}morpholine
ethyl 5-methyl-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(propan-2-yl)-5-[3-(1H-pyrazol-3-yl)phenyl]thiophene-2-carboxamide