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2-(dimethyl-1,3-thiazol-4-yl)-N-[(3S,4R)-4-ethoxyoxolan-3-yl]acetamide
6-fluoro-4-(3-methylpiperidine-1-carbonyl)-2-(1H-pyrazol-4-yl)quinoline
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-one
2-[3-(2,5-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-5-fluoro-N,N-dimethylpyrimidin-4-amine
N-[(1S,2S)-2-(benzyloxy)cyclohexyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
4-(2,6-dimethylpyridin-3-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpyrimidin-2-amine
(2R,6S)-1-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-2,6-dimethylpiperidine
2-{[1-(carbamoylmethyl)piperidin-4-yl]formamido}-2-(3-fluorophenyl)acetic acid
2-{[(4-ethynylphenyl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
4-{4-ethyl-6-[4-(prop-2-en-1-yl)piperazin-1-yl]pyrimidin-2-yl}morpholine
N-methyl-N-(4-methyl-1-phenylpentyl)-2-(pyridin-4-yl)acetamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[(2-methylpyrimidin-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4-{[1-(3-methyloxetane-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
1-(1H-indol-5-yl)-4-methylphthalazine
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
5-[2-(methylsulfanyl)phenoxymethyl]-N-(1-phenylcyclopropyl)-1,2-oxazole-3-carboxamide
(3E)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]hex-3-en-1-one
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
8-(3-aminopropanoyl)-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
dimethyl[3-(3-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}phenoxy)propyl]amine
3-methyl-4-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1,2,5-oxadiazole
1-(2,3-dimethylquinoxalin-6-yl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(propan-2-yl)urea
7-amino-4-(3-chloro-2-fluorophenyl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-2-ylmethyl)pyridin-2-amine
1-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
(3aS,6aS)-2-(1-methyl-1H-indole-3-carbonyl)-5-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
4-[3-(3-hydroxy-3-methylbutyl)benzoyl]-3-(propan-2-yl)piperazin-2-one
2-{3-[(3,4-dimethoxyphenyl)methyl]-5-[(1S)-1-(methylamino)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-6-[1-(propan-2-yl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
2-methyl-6-{1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}pyrimidin-4-ol
1-[2-(piperidin-2-yl)ethyl]-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
7,7-dimethyl-2-[(trimethyl-1H-pyrazol-1-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(3,5-dimethylphenyl)methyl]-4-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]piperazin-2-one
3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propanoic acid
3-acetamido-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
(3aR,6aS)-5-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
1-(4-{[(3S,4R)-3-[(4-ethylpiperazin-1-yl)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
(3S,4S)-1-[(4-chlorophenyl)methyl]-4-(dimethylamino)pyrrolidin-3-ol
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(2-methylnaphthalen-1-yl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[4-(methylamino)pyrimidin-2-yl]-4-(pyrazin-2-yl)-1,4-diazepan-6-ol
1-(ethanesulfonyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
4-(2,4-dichlorophenyl)-2-methylpyrimidine
6-(hydroxymethyl)-N-(2,2,4,4-tetrafluoro-2,4-dihydro-1,3-benzodioxin-6-yl)-1,4-oxazepane-4-carboxamide