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N-(5-chloro-2-methylphenyl)-2-{4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]morpholin-3-yl}acetamide
4-(3,5-dichloro-4-methylbenzoyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
1-(5-fluoro-2-methoxybenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
1-ethyl-5-methyl-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[2-(2-chloro-6-methylphenoxy)ethyl]-2-(propan-2-yloxy)propanamide
N,N-diethyl-4-{[(2-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(5S)-5-({[(3-phenyl-1,2-oxazol-5-yl)methyl](pyridin-2-ylmethyl)amino}methyl)pyrrolidin-2-one
1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-2-(thiophen-2-yl)ethane-1,2-dione
1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)piperazine
3-{2-[({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)carbamoyl)amino]phenyl}-N-methylpropanamide
4-(2,3-dihydro-1H-inden-2-yl)-6-methoxy-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
ethyl 2-(2-{2-[4-(3-phenoxypropanamido)-1H-pyrazol-1-yl]acetamido}ethyl)-1,3-thiazole-4-carboxylate
[(1R,3S,3aS,6aR)-5-benzyl-3-(1-methyl-1H-imidazol-2-yl)-1-(2-methylpropyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methylbenzamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2,5-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]furan-3-carboxamide
(3R,4R)-1-[(2-fluoro-5-methoxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
2-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-N-(5-methyl-1,2-oxazol-3-yl)-2-oxoacetamide
3-(2,6-dimethoxyphenyl)-5-(naphthalen-2-ylmethyl)-1,2,4-oxadiazole
N-(1-cycloheptylpiperidin-3-yl)-1-(furan-2-ylmethyl)piperidine-4-carboxamide
ethyl 1-{[3-cyclohexaneamido-2-(methoxycarbonyl)thieno[2,3-b]pyridin-6-yl]methyl}piperidine-4-carboxylate
3-(aminomethyl)-4-[(2,4-dichlorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
8-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
(1R,5R)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
3-{[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(1,2-oxazol-3-yl)acetamide
1-[(2-chlorophenyl)methyl]-N-[1-(naphthalen-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}methyl)piperidin-2-one
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-methylphenoxy)azetidin-1-yl]butan-1-one
3-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
4-chloro-2-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2,5,6-trimethylpyrimidin-4-amine
2-[4-(4-methoxy-2-methylphenyl)-1H-pyrazol-1-yl]ethan-1-ol
2,5-dimethyl-N-(1-phenylbutyl)furan-3-carboxamide
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
N-[(2S)-1-hydroxypropan-2-yl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(morpholine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(2-methylphenyl)acetamide
3-fluoro-4-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenol
methyl (1S,3S,3aR,6aS)-5-ethyl-1-(hydroxymethyl)-4,6-dioxo-3-(2,4,6-trimethylphenyl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(1-methyl-2-oxoimidazolidine-4-carbonyl)-1-(4-methylphenyl)piperazin-2-one
methyl 3-{1-azabicyclo[3.2.1]octan-5-yloxy}-4-methoxybenzoate
N-(2-hydroxyethyl)-5-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
(1R,5R)-6-[(2,6-difluorophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-ethyl-7-fluoro-N-(pyridin-4-ylmethyl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
N-(1-ethyl-4-methyl-1H-pyrazol-5-yl)-2-[5-(2-methylphenyl)-2H-1,2,3,4-tetrazol-2-yl]acetamide